Anti-cancer activity of capsaicin and its analogs in gynecological cancers
KC Brown, AM Sugrue, KB Conley… - … in cancer research, 2024 - pubmed.ncbi.nlm.nih.gov
Capsaicin is the hot and pungent ingredient of chili peppers. It is a potent pain-relieving
agent and is often present in over-the-counter analgesic lotions and creams. Several …
agent and is often present in over-the-counter analgesic lotions and creams. Several …
[HTML][HTML] Capsaicin Exerts Antitumor Activity in Mesothelioma Cells
E Andretta, A Costa, E Ventura, M Quintiliani… - Nutrients, 2024 - mdpi.com
Background/Objectives: Mesothelioma is an aggressive cancer with limited treatment
options. Mesothelioma therapy often involves a multimodal approach including surgery …
options. Mesothelioma therapy often involves a multimodal approach including surgery …
Development and Evaluation of Bis-benzothiazoles as a New Class of Benzothiazoles Targeting DprE1 as Antitubercular Agents
Benzothiazole-bearing compounds have emerged as potential noncovalent DprE1 (
decaprenylphosphoryl-β-d-ribose-2′-epimerase) inhibitors active against Mycobacterium …
decaprenylphosphoryl-β-d-ribose-2′-epimerase) inhibitors active against Mycobacterium …
Capsaicin derivatives: Synthesis and biological activity
S Liu, X Zheng, J Wu, Y Zeng, X Wei… - Chemical Biology & …, 2024 - Wiley Online Library
Capsaicin is the main active ingredient of chili peppers and the most pungent alkaloid. It is
reported that capsaicin has many pharmacological effects such as analgesia, anticancer …
reported that capsaicin has many pharmacological effects such as analgesia, anticancer …
Piperazine-1, 2, 3-triazole scaffolds: design, synthesis, anticancer and antimicrobial evaluation
P Yadav, CP Kaushik, A Yadav, J Yadav… - Future Medicinal …, 2023 - Taylor & Francis
Aim: The objective of the present study is to design and synthesize diverse piperazine-1, 2, 3-
triazole scaffolds as key pharmacophores possessing antimicrobial/anticancer activities …
triazole scaffolds as key pharmacophores possessing antimicrobial/anticancer activities …
[HTML][HTML] Synthesis of new 1, 2, 3-triazole linked benzimidazolidinone: Single crystal X-ray structure, biological activities evaluation and molecular docking studies
H Al-Ghulikah, A Ghabi, H Mtiraoui, E Jeanneau… - Arabian Journal of …, 2023 - Elsevier
Abstract A novel series of 1, 2, 3-triazole-benzimidazolidinone hybrid derivatives were
designed and synthesized via click reaction, between various aryl azide and a terminal …
designed and synthesized via click reaction, between various aryl azide and a terminal …
Flow Synthesis of Capsaicin and Capsaicinoid Analogues
MJ Orosz, B Rávai, B Mátravölgyi… - … Sustainable Chemistry & …, 2024 - ACS Publications
Capsaicin and its derivatives are special alkaloids responsible for the pungency of spicy
pepper fruits and are mainly used in the pharmaceutical, food, and cosmetic industries. Until …
pepper fruits and are mainly used in the pharmaceutical, food, and cosmetic industries. Until …
Small Peptide Conjugates of Benzothiazole‐2‐Carboxylic Acids Targeting DprE1 Against Tuberculosis
Inhibitors of Decaprenylphosphoryl‐β‐D‐ribose 2′‐epimerase (DprE1) are being
thoroughly explored as potential pharmacological entities for the development of new anti …
thoroughly explored as potential pharmacological entities for the development of new anti …
Synthesis of New Imidazo [1, 2‐a] pyridine Triazole Hybrid Molecules as Potential Apoptotic Antitumor Agents
Abstract Novel imidazo [1, 2‐a] pyridines bearing 1, 2, 3‐triazole moieties at the C3 position
were synthesized. After the characterization of the synthesized compounds, their in vitro …
were synthesized. After the characterization of the synthesized compounds, their in vitro …