In the past decades, the iridium-catalyzed C–H bond borylation and other newly discovered
catalytic borylation reactions have received extensive research interests and developed into …

The iridium‐catalysed borylation of aromatic C− H bonds has become the preferred method
for the synthesis of aromatic organoboron compounds. The reaction is highly efficient …

Indazoles are a very important class of N‐containing heterocycles with a wide range of
biological and medicinal properties. The presence of different functionalities on indazole …

In the absence of a steric directing group, iridium-catalyzed C–H borylation of N-protected
indazoles occurs rapidly and selectively at C-3 and the resulting boronate esters can be …

The palladium‐catalyzed direct arylation of 2 H‐indazoles with aryl bromides for the
preparation of 3‐aryl‐2 H‐indazoles was found to proceed in high yields when using only …

The indazole system was found in various biologically active molecules. For very recent
applications, indazole was reported as eg, selective estrogen receptor degraders, 1 …

This report highlights the recent advances in direct C–H bond functionalization of 5, 5-and 6,
5-fused heterocycles containing at least two nitrogen atoms. Besides C–C bond formation, C …

Abstract Die Ir‐katalysierte Borylierung aromatischer C‐H‐Bindungen ist heute die
bevorzugte Methode zur Synthese aromatischer Organoborverbindungen. Sie ist …

A series of 3-aryl indazoles and 1-methyl-3-aryl indazole derivatives are prepared with
exceptional yields by coupling with several arylboronic acids and methylation by two …

The C3 direct arylation of 1 H-indazole and 1 H-7-azaindazole has been a significant
challenge due to the lack of the reactivity at this position. In this paper, we describe a mild …