Diboron (4) compounds: from structural curiosity to synthetic workhorse

EC Neeve, SJ Geier, IAI Mkhalid, SA Westcott… - Chemical …, 2016 - ACS Publications
Although known for over 90 years, only in the past two decades has the chemistry of diboron
(4) compounds been extensively explored. Many interesting structural features and reaction …

Performances of symmetrical achiral ferrocenylphosphine ligands in palladium-catalyzed cross-coupling reactions: A review of syntheses, catalytic applications and …

A Fihri, P Meunier, JC Hierso - Coordination Chemistry Reviews, 2007 - Elsevier
Ferrocene derivatives bearing donor atoms led to the generation of several classes of
metallo-ligands, which collectively show an impressive diversity of applications, especially in …

Glucopyranosyl-substituted phenyl derivatives, medicaments containing such compounds, their use and process for their manufacture

M Eckhardt, P Eickelmann, F Himmelsbach… - US Patent …, 2009 - Google Patents
Glucopyranosyl-substituted benzene derivatives of general formula I where the groups R* to
R* as well as R7, R”, R7 are defined herein and the tautomers, the stereoisomers thereof …

Recent Advances on Amino Acid Modifications via C–H Functionalization and Decarboxylative Functionalization Strategies

S Mondal, S Chowdhury - Advanced Synthesis & Catalysis, 2018 - Wiley Online Library
Over the recent decade tremendous interest has been developed on the synthetic
modification of natural as well as non‐proteinogenic amino acids and non‐natural linkages …

Palladium-and copper-catalyzed synthesis of medium-and large-sized ring-fused dihydroazaphenanthrenes and 1, 4-benzodiazepine-2, 5-diones. Control of reaction …

G Cuny, M Bois-Choussy, J Zhu - Journal of the American …, 2004 - ACS Publications
Methods for the synthesis of dihydroazaphenanthrene fused to macrocycles (2) and medium-
ring heterocycles (4), as well as 1, 4-benzodiazepine-2, 5-diones (5), are developed. A …

The Suzuki–Miyaura cross-coupling as a versatile tool for peptide diversification and cyclization

T Willemse, W Schepens, HWT van Vlijmen… - Catalysts, 2017 - mdpi.com
The (site-selective) derivatization of amino acids and peptides represents an attractive field
with potential applications in the establishment of structure–activity relationships and …

Synthesis of chromeno [3, 4-b] indoles as Lamellarin D analogues: A novel DYRK1A inhibitor class

C Neagoie, E Vedrenne, F Buron, JY Mérour… - European journal of …, 2012 - Elsevier
A library of substituted chromeno [3, 4-b] indoles was developed as Lamellarin isosters.
Synthesis was achieved from indoles after a four-step pathway sequence involving C-3 …

Pharmaceutical composition comprising a glucopyranosyl-substituted benzene derivate

K Dugi, M Mark, L Thomas, F Himmelsbach - US Patent 8,551,957, 2013 - Google Patents
The invention relates to a pharmaceutical composition according to the claim 1 comprising a
glucopyranosyl-Sub stituted benzene derivative in combination with a DPP IV inhibitor which …

Synthesis of the side chain cross-linked tyrosine oligomers dityrosine, trityrosine, and pulcherosine

O Skaff, KA Jolliffe, CA Hutton - The Journal of organic chemistry, 2005 - ACS Publications
An efficient synthesis of dityrosine and the first syntheses of the tyrosine trimers trityrosine
and pulcherosine have been achieved. Protected 3-iodotyrosine underwent tandem Miyaura …

Crystalline form of 1-chloro-4-(β-D-glucopyranos-1-yl)-2-[4-((S)-tetrahydrofuran-3-yloxy)-benzyl]-benzene, a method for its preparation and the use thereof for …

F Himmelsbach, S Schmid, M Schuehle… - US Patent …, 2010 - Google Patents
US7713938B2 - Crystalline form of 1-chloro-4-(β-D-glucopyranos-1-yl)-2-[4-((S)-tetrahydrofuran-3-yloxy)-benzyl]-benzene,
a method for its preparation and the use thereof for preparing medicaments - Google …