Microwave-assisted synthesis of nitrogen-containing heterocycles

A Majumder, R Gupta, A Jain - Green Chemistry Letters and …, 2013 - Taylor & Francis
In the recent years, microwave (MW) radiation is widely used as a source of heating in
organic synthesis. Since the discovery of the MW heating approach, MW-assisted reaction …

2-(2-Arylphenyl) benzoxazole as a novel anti-inflammatory scaffold: synthesis and biological evaluation

K Seth, SK Garg, R Kumar, P Purohit… - ACS medicinal …, 2014 - ACS Publications
The 2-(2-arylphenyl) benzoxazole moiety has been found to be a new and selective ligand
for the enzyme cyclooxygenase-2 (COX-2). The 2-(2-arylphenyl) benzoxazoles 3a–m have …

Palladium catalyzed C sp2–H activation for direct aryl hydroxylation: the unprecedented role of 1, 4-dioxane as a source of hydroxyl radicals

K Seth, M Nautiyal, P Purohit, N Parikh… - Chemical …, 2015 - pubs.rsc.org
A novel strategy for direct aryl hydroxylation via Pd-catalysed Csp2–H activation through an
unprecedented hydroxyl radical transfer from 1, 4-dioxane, used as a solvent, is reported …

C‐N and N‐N bond formation via Reductive Cyclization: Progress in Cadogan/Cadogan‐Sundberg Reactionǂ

M Kaur, R Kumar - ChemistrySelect, 2018 - Wiley Online Library
Abstract Cadogan/Cadogan‐Sundberg cyclization reaction has been reported as one of the
most efficient routes for the synthesis of a wide variety of N‐heterocycles from the easily …

Efficient protocol for the synthesis of quinoxaline, benzoxazole and benzimidazole derivatives using glycerol as green solvent

HM Bachhav, SB Bhagat, VN Telvekar - Tetrahedron Letters, 2011 - Elsevier
A straightforward, efficient and more sustainable catalyst-free method has been developed
for the synthesis of quinoxaline, benzoxazole, and benzimidazole ring system in glycerol to …

Convenient synthesis of 2, 3-disubstituted quinazolin-4 (3 H)-ones and 2-styryl-3-substituted quinazolin-4 (3 H)-ones: Applications towards the synthesis of drugs

D Kumar, PS Jadhavar, M Nautiyal, H Sharma… - RSC Advances, 2015 - pubs.rsc.org
Simple, convenient, and green synthetic protocols have been developed for the one pot
synthesis of 2, 3-disubstituted quinazolin-4 (3H)-ones and 2-styryl-3-substituted quinazolin-4 …

Green synthesis of novel pyridines via one-pot multicomponent reaction and their anti-inflammatory evaluation

HM Abd El-Lateef, AA Abdelhamid, MM Khalaf… - ACS …, 2023 - ACS Publications
A functional and environmentally green procedure for the design of novel pyridine 5a–h and
7a–d derivatives through two pathways is presented. The first pathway is via a one-pot, four …

Benzimidazoquinazolines as new potent anti-TB chemotypes: Design, synthesis, and biological evaluation

PS Jadhavar, KI Patel, TM Dhameliya, N Saha… - Bioorganic …, 2020 - Elsevier
In search for new molecular entities as anti-TB agents, the benzimidazoquinazoline
polyheterocyclic scaffold has been designed adopting the scaffold hopping strategy. Thirty …

Cu-Nanoparticles: efficient catalysts for the oxidative cyclization of Schiffs' bases

M Kidwai, V Bansal, A Saxena, S Aerry, S Mozumdar - Tetrahedron letters, 2006 - Elsevier
Cu-Nanoparticles provide an efficient catalysis for the synthesis of 2-arylbenzoxazoles by
the coupling of aromatic or heteroaromatic aldehydes with 2-aminophenol though the …

Facile and efficient one‐pot protocol for the synthesis of benzoxazole and benzothiazole derivatives using molecular iodine as catalyst

F Matloubi Moghaddam… - Synthetic …, 2006 - Taylor & Francis
Rapid and efficient condensation reactions of 2‐aminothiophenol and 2‐aminophenol with
various aldehydes were carried out using I2 in solvent‐free conditions with or without …