The purpose of this review is to highlight ten years of success in the synthesis of six-
membered N-heterocycles using alkynes and nitrogen sources as substrates. It is our hope …

The synthesis of quinoline derivatives through multicomponent reactions (MCRs) has
emerged as an efficient and versatile strategy in organic synthesis. MCRs offer the …

In this paper, we report the synthesis of alkyl-tethered alkynes through ozone-mediated and
FeII-catalyzed dealkenylative alkynylation of unactivated alkenes in the presence of alkynyl …

A copper-catalyzed protocol for the construction of various 2-aryl (alkyl)-3-acylquinolines or
3-arylquinolines using readily available anthranils and 1, 3-diketones or aldehydes as …

An efficient one-pot synthesis of 4-(1 H)-quinolones through an orthogonal engagement of
diverse o-haloaryl ynones with ammonia in the presence of Cu (I), involving tandem Michael …

A novel palladium-catalyzed protocol for the synthesis of 2-arylquinolines via tandem
reaction of 2-aminostyryl nitriles with arylboronic acids has been developed with good …

A [4+ 2] annulation involving cascade Knoevenagel, aza-Wittig and dehydrofluorination
reactions is developed for the synthesis of substituted quinolin-4-ols including analogs …

A novel Cu-catalyzed tandem C–N and C–C bond-formation reaction has been developed
to furnish 2-substituted-4-(1H)-quinolones. 4-(1H)-quinolones play an important role in …

A method for the catalyst-free synthesis of pyrroloquinolinediones and
quinolinedicarboxylates is developed through a one-pot synthesis involving denitrogenation …

A Rh (III)-catalyzed carboamination of alkynyl cycloalkanols with arylamines has been
developed. This transformation involves a novel Csp2–H/Csp3–Csp3 activation relay and …