Implementation of diverse synthetic and strategic approaches to biologically active sulfamides

JJ Jun, XQ Xie - ChemistrySelect, 2021 - Wiley Online Library
Sulfamide compounds are an important class of motif in various applications in
pharmaceutical agents, agriculture, and material science. In this review, various synthetic …

Synthesis and antibacterial activity of sulfonamides. SAR and DFT studies

W Boufas, N Dupont, M Berredjem, K Berrezag… - Journal of Molecular …, 2014 - Elsevier
A series of substituted sulfonamide derivatives were synthesized from chlorosulfonyl
isocyanate (CSI) in tree steps (carbamoylation, sulfamoylation and deprotection) …

Preparation and uses of chlorinated glycerol derivatives

A Canela-Xandri, M Balcells, G Villorbina, P Christou… - Molecules, 2020 - mdpi.com
Crude glycerol (C3H8O3) is a major by-product of biodiesel production from vegetable oils
and animal fats. The increased biodiesel production in the last two decades has forced …

A one-pot three-component synthesis of novel α-sulfamidophosphonates under ultrasound irradiation and catalyst-free conditions

B Belhani, M Berredjem, M Le Borgne, Z Bouaziz… - RSC Advances, 2015 - pubs.rsc.org
An efficient and convenient one-pot synthesis of novel α-sulfamidophosphonates is
described via a three-component reaction. This reaction was carried out through a three …

Novel α-sulfamidophosphonate analogues of fotemustine: efficient synthesis using ultrasound under solvent-free conditions

M Guerfi, M Berredjem, A Bouzina… - Monatshefte für Chemie …, 2020 - Springer
The development of new clean and effective processes for the preparation of new
elaborated compounds is currently an important research axis in organic chemistry, thus in …

A simple and eco-sustainable method for the sulfonylation of amines under microwave-assisted solvent-free conditions

S Lakrout, H K'tir, A Amira, M Berredjem, NE Aouf - RSC Advances, 2014 - pubs.rsc.org
A new environmentally benign, simple, and efficient protocol for the chemoselective
sulfonylation of various structural amines using microwave irradiation under solvent-and …

One-pot synthesis of novel oxazaphosphinanes under ultrasound irradiation and solvent-free conditions

B Belhani, A Bouzina, M Berredjem, N Aouf - Monatshefte für Chemie …, 2015 - Springer
A rapid and efficient solvent-free one-pot synthesis of novel oxazaphosphinane is described
under ultrasound irradiation. This reaction was carried out through a three-component …

Synthesis, in silico study (DFT, ADMET) and crystal structure of novel sulfamoyloxy-oxazolidinones: Interaction with SARS-CoV-2

A Bouzina, M Berredjem, S Bouacida, K Bachari… - Journal of Molecular …, 2022 - Elsevier
A new series of sulfamoyloxyoxazolidinone (SOO) derivatives have been synthesized and
characterized by single-crystal X-ray diffraction, NMR, IR, MS and EA. Chemical reactivity …

Efficient Synthesis, Characterization, and Antibacterial Activity of Novel N-Acylsulfonamides and Sulfonylureas

C Hadjer, B Malika, B Wahida, B Fouzia… - … , Sulfur, and Silicon …, 2014 - Taylor & Francis
A series of novel sulfonylureas and N-acylsulfonamides derivatives were synthesized and
characterized by 1H NMR, 13C NMR, and HRMS. These compounds were synthesized …

An efficient synthesis, characterization, DFT study and molecular docking of novel sulfonylcycloureas

M Guerfi, M Berredjem, R Bahadi, SE Djouad… - Journal of molecular …, 2021 - Elsevier
Abstract Sulfonylcycloureas derivatives (3a-3e) are novel heterocyclic compounds
synthesized by condensation reaction of several sulfonamides derived from aminoesters (1a …