Antibacterial-resistance speaks to an overall alarm, particularly in regards to the flare-up of
methicillin-resistance Staphylococcus aureus (MRSA), a classic reason for genuine skin and …

The extraordinary impact of metal-based complexes on synthetic methods is still recognized
nowadays, and attempts are currently undertaken to further extend the use of metal-assisted …

Over the last two decades, transition-metal catalyzed C–H functionalization of indoles has
emerged as an area of extensive research and tremendous progress has been made in this …

A series of new indole-2-carboxylic acid derived mono and bis 1, 4-disubstituted 1, 2, 3
triazoles (I 1–I 6 and I 7–I 12) were synthesized and screened for their anticancer (in vitro …

Herein, we describe an efficient transition-metal-free regioselective C3alkylation of indoles
for the synthesis of bis (indolyl) methanes and 3-styryl indoles. Nitrobenzene is employed as …

Herein is reported the first asymmetric utilization of aryldiazonium cations as a source of
electrophilic nitrogen. This is achieved through a chiral anion phase‐transfer …

A mild and selective C–H arylation strategy for indoles, benzofurans and benzothiophenes
is described. The arylation method engages aryldiazonium salts as arylating reagents in …

A dual vicinal functionalisation cascade involving the union of heterocycles and allyl
sulfoxides is described. In particular, the approach provides efficient one-step access to …

A new approach to C-2 arylated indoles has been developed by utilizing a ruthenium-
catalyzed, heteroatom-directed regioselective C–H arylation. The reaction is highly site …

A halogen-atom-transfer (XAT)-based method for carbonylazotization of pyrroles or indoles
with aryldiazonium salts and polyhalomethanes via dual C (sp2)–H bond functionalization is …