Acetamides: chemotherapeutic agents for inflammation-associated cancers
Now clear evidences are available to support the hypothesis that inflammation accelerates
the conditions including events and molecules that reach to various types of cancers …
the conditions including events and molecules that reach to various types of cancers …
Immunostimulatory and antagonistic potential of the methanolic extract of Oedogonium intermedium SCB in Cirrhinus reba challenged with Aeromonas hydrophila
S Chattaraj, PK Das Mohapatra - Aquaculture International, 2024 - Springer
Studies on antimicrobial and immunotherapeutic agents have become a priority in the
management of fish ailments. The Reba carp (Cirrhinus reba) is currently passing through a …
management of fish ailments. The Reba carp (Cirrhinus reba) is currently passing through a …
Antimycobacterial, Molecular Docking and ADME Studies of Spiro Naphthyridine Pyrimidine and N‐(Quinolin‐8‐yl) acetamide Derivatives
S Satisha, VG Revanasiddappa, S Ramaiah - ChemistrySelect, 2023 - Wiley Online Library
Two series of compounds viz., spiro naphthyridine pyrimidine derivatives and N‐(quinolin‐8‐
yl) acetamide derivatives which possess the quinoline core moiety were designed and …
yl) acetamide derivatives which possess the quinoline core moiety were designed and …
Novel quercetin and apigenin-acetamide derivatives: design, synthesis, characterization, biological evaluation and molecular docking studies
Flavonoids exhibit essential but limited biological properties which can be enhanced
through chemical modifications. In this study, we designed, synthesized, and characterized …
through chemical modifications. In this study, we designed, synthesized, and characterized …
[HTML][HTML] Design, synthesis, molecular docking and biological evaluation of imides, pyridazines, and imidazoles derived from itaconic anhydride for potential …
New functionalized N-heterocyclic derivatives were synthesized from an itaconic anhydride
(ITA) precursor and characterized by spectral and analytical data. All of the synthesized …
(ITA) precursor and characterized by spectral and analytical data. All of the synthesized …
Design and synthesis of aminothiazole-benzazole based amide: antiproliferative, antimigration activity and molecular docking studies
In this study, we synthesized a series of amide-functionalized aminothiazole-benzazole
analogs for potential application in cancer treatment. The chemical structures of these …
analogs for potential application in cancer treatment. The chemical structures of these …
Synthesis and bioactivity evaluation of novel acetamide-derived compounds bearing a methylsulfonyl unit
P Li, Z Wang, L Yu - Phosphorus, Sulfur, and Silicon and the …, 2024 - Taylor & Francis
This study reports the synthesis and structural characterization of a series of novel
acetamide-derived compounds containing a methylsulfonyl unit. The in vitro antibacterial …
acetamide-derived compounds containing a methylsulfonyl unit. The in vitro antibacterial …
Synthesis, molecular docking and biological evaluation of novel bis-pyrazole derivatives for analgesic, anti-inflammatory and antimicrobial activities
PS Nayak, B Narayana, BK Sarojini, J Fernades… - Medicinal Chemistry …, 2015 - Springer
A new series of bis-pyrazoles were synthesized by Michael addition of hydrazine to
chalcones. The starting-material-substituted acetophenones required for the synthesis of …
chalcones. The starting-material-substituted acetophenones required for the synthesis of …
Synthesis of Small Molecule Library of Novel Nicotinamide Derivatives as Anticancer Agents and Computational Screening
RM Malothu, G Thalari - ChemistrySelect, 2025 - Wiley Online Library
A small molecule library of nicotinamide derivatives synthesized and characterized their
structure by interpretation of 1H NMR, 13C NMR, and Mass spectral data. The new …
structure by interpretation of 1H NMR, 13C NMR, and Mass spectral data. The new …
Potent pharmacophoric aminothiazole derivatives as FabH inhibitors for antibacterial activity: in vitro and in silico approach
The present work reports the design, synthesis, characterization and antibacterial screening
of novel aminothiazole derivatives as FabH inhibitor [β-ketoacyl-ACP synthase (KAS)] which …
of novel aminothiazole derivatives as FabH inhibitor [β-ketoacyl-ACP synthase (KAS)] which …