Design and environmentally benign synthesis of novel thiophene appended pyrazole analogues as anti-inflammatory and radical scavenging agents: Crystallographic …

MG Prabhudeva, S Bharath, AD Kumar, S Naveen… - Bioorganic …, 2017 - Elsevier
Oxidative-stress induces inflammatory diseases and infections caused by drug-resistant
microbial strains are on the rise necessitating the discovery of novel small-molecules for …

Synthesis, crystal structure and Hirshfeld surface analysis of 5-(3, 4-dimethoxyphenyl)-3-(thiophen-2-yl)-4, 5-dihydro-1H-pyrazole-1-carboxamide

M Prabhuswamy, K Kumara, G Pavithra… - Chemical Data …, 2016 - Elsevier
Abstract The compound, 5-(3, 4-Dimethoxyphenyl)-3-(thiophen-2-yl)-4, 5-dihydro-1H-
pyrazole-1-carboxamide was synthesized by the reaction of 3-(3, 4-dimethoxyphenyl)-1 …

[HTML][HTML] 4-(Thiophen-2-yl)-2-[4-(trifluoromethyl) phenyl]-2, 3-dihydro-1, 5-benzothiazepine

BC Manjunath, M Manjula… - … Section E: Structure …, 2014 - scripts.iucr.org
In the title compound, C20H14F3NS2, the seven-membered thiazepine ring adopts a slightly
distorted twist–boat conformation. The mean plane of the five-membered thiophene ring …

[PDF][PDF] Synthesis of novel 1, 4-benzothiazepines and in vitro screening of their antimicrobial activity

KR Raghavendra, KA Kumar… - Int. J. Pharm. Pharm …, 2014 - researchgate.net
Objective: In search of new potential antimicrobial agents, the aim of the present study was
synthesize the series of 1, 4-Benzothiazepine analogs by a simple and accessible approach …

[PDF][PDF] 2-(3, 4-Dimethoxyphenyl)-4-(thiophen-2-yl)-2, 3-dihydro-1, 5-benzothiazepine

BC Manjunath, M Manjula… - … Section E: Structure …, 2014 - journals.iucr.org
In the title compound, C21H19NO2S2, the seven-membered thiazepine ring adopts a
slightly distorted twist boat conformation. The dihedral angle between the benzene rings is …

Synthesis, crystal and molecular structure, and antimicrobial activity of ethyl 2-(4-methylbenzylidene)-3-oxobutanoate

AK Kariyappa, N Shivalingegowda, DK Achutha… - Chemical Data …, 2016 - Elsevier
Abstract Ethyl 2-(4-methylbenzylidene)-3-oxobutanoate was synthesized by Knoevenagel
condensation reaction of 4-methylbenzaldehyde and ethyl acetoacetate in the presence of …

[PDF][PDF] An easy route to synthesis of thiophene tagged pyrimidin-2-thiones as antibacterial agents

VK Shruthi, CB Vagish… - Journal of Chemical and …, 2015 - researchgate.net
ABSTRACT A series of substituted pyrimidin-2-thiones tagged with thiophene moiety was
synthesized by an easy procedure. The reaction of chalcones 1-5 and thiourea 6 in the …

[PDF][PDF] An efficient route to synthesis of pyrazoline carboxamides bearing thiophene moiety as antimicrobial agents

SP Vijaychand, G Pavithra, KR Raghavendra… - Der Pharma …, 2015 - researchgate.net
ABSTRACT A series of new pyrazoline carbothioamides bearing thiophene moiety were
synthesized by simple one pot procedure. The cyclocondensation reaction of chalcones 1a …

Synthesis and antifungal activity of novel pyrimidin-2-one analogues

G Shwetha Hegde, A Dileep Kumar… - Journal of Chemical …, 2015 - eprints.uni-mysore.ac.in
A series of thiophene appended substituted pyrimidin-2-one analogues were synthesized by
an accessible approach. The reaction of chalcones 1 (ae) and urea 2 in the presence …

[PDF][PDF] Synthesis and Antifungal Potency of Novel 4-Aryl-2-(2, 4-Dichlorophenyl)-1, 4-Benzothiazepine Derivatives

DM Shyam, KA Kumar, HP Jayadevappa - researchgate.net
An easy procedure for the synthesis of 1, 4-benzothiazepines was described. The reaction of
chalcones, 1a-g and 2-aminothiophenol, 2 in the presence of catalytic amount of …