A patent review on the current developments of benzoxazoles in drug discovery
The benzoxazole moiety is widely found in various natural compounds, which are often
found to be biologically active. Due to its versatile biological properties, benzoxazole has …
found to be biologically active. Due to its versatile biological properties, benzoxazole has …
A Review on Five and Six-Membered Heterocyclic Compounds Targeting the Penicillin-Binding Protein 2 (PBP2A) of Methicillin-Resistant Staphylococcus aureus …
Staphylococcus aureus is a common human pathogen. Methicillin-resistant Staphylococcus
aureus (MRSA) infections pose significant and challenging therapeutic difficulties. MRSA …
aureus (MRSA) infections pose significant and challenging therapeutic difficulties. MRSA …
Synthesis, molecular docking, molecular dynamics, DFT and antimicrobial activity studies of 5-substituted-2-(p-methylphenyl) benzoxazole derivatives
Abstract In this study, new 2-(p-methylphenyl)-5-(2-substitutedacetamido) benzoxazole
derivatives were synthesized, and antimicrobial activities on six bacteria and their twelve …
derivatives were synthesized, and antimicrobial activities on six bacteria and their twelve …
Antimicrobial and antiproliferative activity studies of some new quinoline-3-carbaldehyde hydrazone derivatives
In this study, a total of 22 piece quinoline-3-carbaldehyde hydrazone derivative compounds
were designed and synthesized, 2 of which were not original, their antimicrobial activities …
were designed and synthesized, 2 of which were not original, their antimicrobial activities …
An efficient synthesis of novel di-heterocyclic benzazole derivatives and evaluation of their antiproliferative activities
A series of unsymmetrical nine di-heterocyclic compounds of benzazole derivatives were
synthesized at one step via cyclization reaction. The compounds evaluated for in vitro …
synthesized at one step via cyclization reaction. The compounds evaluated for in vitro …
Alternative benzoxazole assembly discovered in anaerobic bacteria provides access to privileged heterocyclic scaffold
T Horch, EM Molloy, F Bredy, VG Haensch… - Angewandte …, 2022 - Wiley Online Library
Benzoxazole scaffolds feature prominently in diverse synthetic and natural product‐derived
pharmaceuticals. Our understanding of their bacterial biosynthesis is, however, limited to …
pharmaceuticals. Our understanding of their bacterial biosynthesis is, however, limited to …
[PDF][PDF] Design, synthesis, antimicrobial and anticancer activity of some novel benzoxazole-isatin conjugates
E Susithra, S Rajkumar… - … Res. Appl. Chem, 2022 - biointerfaceresearch.com
A series of novel benzoxazole-isatin conjugates were synthesized by treating 2-amino
benzoxazole with 5 and 7 substituted isatin derivatives and were screened for in vitro …
benzoxazole with 5 and 7 substituted isatin derivatives and were screened for in vitro …
Synthesis, molecular docking, and DFT studies of some new 2, 5-disubstituted benzoxazoles as potential antimicrobial and cytotoxic agents
In this study, a total of 17 piece 2, 5-disubstituted benzoxazole derivatives were synthesized,
2 of which were not original, their antimicrobial activities were determined using …
2 of which were not original, their antimicrobial activities were determined using …
Synthesis, quantum mechanical calculations, antimicrobial activities and molecular docking studies of five novel 2, 5-disubstituted benzoxazole derivatives
In this study, five new 2-(p-(Substituted) phenyl)-5-(3-(4-ethylpiperazine-1-yl) propionamido)
benzoxazole derivatives (B7-B11) were designed, synthesized, and their antimicrobial …
benzoxazole derivatives (B7-B11) were designed, synthesized, and their antimicrobial …
Bisbenzoxazole Derivatives: Design, Synthesis, in Vitro Antimicrobial, Antiproliferative Activity, and Molecular Docking Studies
Four series of bisbenzoxazole derivatives were designed, synthesized, and screened for
antiproliferative and antimicrobial activities. Generally, all synthesized bisbenzoxazoles (9 …
antiproliferative and antimicrobial activities. Generally, all synthesized bisbenzoxazoles (9 …