Past, present and future of the Biginelli reaction: a critical perspective.

JS Sandhu - ARKIVOC: Online Journal of Organic …, 2012 - search.ebscohost.com
This review covers up to 2010 and some available references of 2011 of synthetic advances
in the Biginelli reaction, including recent mechanistic advances, new building blocks, new …

Biginelli reaction: Polymer supported catalytic approaches

RV Patil, JU Chavan, DS Dalal, VS Shinde… - ACS combinatorial …, 2019 - ACS Publications
The Biginelli product, dihydropyrimidinone (DHPM) core, and its derivatives are of immense
biological importance. There are several methods reported as modifications to the original …

A chemical placebo: NaCl as an effective, cheapest, non-acidic and greener catalyst for Biginelli-type 3,4-dihydropyrimidin-2(1H)-ones (-thiones) synthesis

MA Kolosov, VD Orlov, DA Beloborodov… - Molecular diversity, 2009 - Springer
Despite prior reports of several really effective catalytic and non-catalytic approaches
towards Biginelli's 3, 4-dihydropyrimidin-2 (1 H)-ones, an overwhelming number of new …

Design, ecofriendly synthesis, anticancer and antimicrobial screening of innovative Biginelli dihydropyrimidines using β-aroylpyruvates as synthons

A El-Malah, Z Mahmoud, H Hamed Salem… - … Chemistry Letters and …, 2021 - Taylor & Francis
New ecofriendly Biginelli reaction procedures have been adapted to prepare new
dihydropyrimidines (DHPMs) using a multicomponent one-pot reaction. All the synthesized …

Dowex-50W promoted synthesis of 14-aryl-14H-dibenzo [a, j] xanthene and 1, 8-dioxo-octahydroxanthene derivatives under solvent-free conditions

GI Shakibaei, P Mirzaei, A Bazgir - Applied Catalysis A: General, 2007 - Elsevier
Dowex-50W promoted synthesis of 14-aryl-14H-dibenzo[a,j]xanthene and 1,8-dioxo-octahydroxanthene
derivatives under solvent-free conditions - ScienceDirect Skip to main contentSkip to article …

Microwave-induced bismuth nitrate-catalyzed synthesis of dihydropyrimidones via Biginelli condensation under solventless conditions

BK Banik, AT Reddy, A Datta, C Mukhopadhyay - Tetrahedron Letters, 2007 - Elsevier
Microwave-induced bismuth nitrate-catalyzed synthesis of dihydropyrimidones via Biginelli
condensation under solventless conditions - ScienceDirect Skip to main contentSkip to article …

New potential of the classical Biginelli reaction

SV Vdovina, VA Mamedov - Russian Chemical Reviews, 2008 - iopscience.iop.org
The published data on the Biginelli reaction are generalised and systematised. The major
attention is focused on the publications of the last seven years. Possible reaction …

Pyrimidine-based antimalarials: design strategies and antiplasmodial effects

K Singh, T Kaur - MedChemComm, 2016 - pubs.rsc.org
Pyrimidine-containing compounds have attracted great attention because of their biological
effects, therapeutic potential and flexibility in structural modification by way of diversifying …

Design, Synthesis and Antiviral Potential of 14-Aryl/Heteroaryl-14H-dibenzo[a,j]xanthenes Using an Efficient Polymer-Supported Catalyst

K Reddi Mohan Naidu, B Satheesh Krishna… - Molecules, 2012 - mdpi.com
Polyethyleneglycol bound sulfonic acid (PEG-OSO3H), a chlorosulphonic acid-modified
polyethylene glycol was successfully used as an efficient and eco-friendly polymeric catalyst …

Organocatalytic application of ionic liquids:[bmim][MeSO4] as a recyclable organocatalyst in the multicomponent reaction for the preparation of dihydropyrimidinones …

SR Roy, PS Jadhavar, K Seth, KK Sharma… - …, 2011 - thieme-connect.com
The organocatalytic potential of 1-butyl-3-methylimidazolium-based room-temperature ionic
liquids has been investigated for the synthesis of dihydropyrimidinones and-thiones by a …