Asymmetric phosphoric acid–catalyzed four-component Ugi reaction
INTRODUCTION The four-component Ugi reaction (Ugi-4CR) assembles peptide-like α-
acylaminoamides through one-pot reaction of a carbonyl compound, an amine, an acid, and …
acylaminoamides through one-pot reaction of a carbonyl compound, an amine, an acid, and …
Metabolic inhibitors of bacterial glycan biosynthesis
The bacterial cell wall is a quintessential drug target due to its critical role in colonization of
the host, pathogen survival, and immune evasion. The dense cell wall glycocalyx contains …
the host, pathogen survival, and immune evasion. The dense cell wall glycocalyx contains …
Enantioselective [4+ 2]-annulation of azlactones with copper-allenylidenes under cooperative catalysis: synthesis of α-quaternary α-acylaminoamides
AK Simlandy, B Ghosh, S Mukherjee - Organic letters, 2019 - ACS Publications
The first enantioselective decarboxylative [4+ 2]-annulation of ethynyl benzoxazinanones
with azlactones has been developed under cooperative copper and bifunctional tertiary …
with azlactones has been developed under cooperative copper and bifunctional tertiary …
Novel diamide derivatives: Synthesis, characterization, urease inhibition, antioxidant, antibacterial, and molecular docking studies
Ş Çakmak - Journal of Molecular Structure, 2022 - Elsevier
Novel diamides (I-VI) were synthesized, corroborated by various spectroscopic techniques
including IR, 1 H NMR, 13 C NMR, mass spectrophotometry and elemental analysis. The in …
including IR, 1 H NMR, 13 C NMR, mass spectrophotometry and elemental analysis. The in …
A new type of heterogeneous catalysis strategy for organic reactions: Ugi-3CR catalyzed by highly stable MOFs with exposed carboxyl groups
J Liu, Y Li, N Liu, N Huang, L Wang, D Li - Organic Chemistry Frontiers, 2022 - pubs.rsc.org
A mild, highly efficient, and simple Ugi-3CR using a novel organic framework material Cu-
COOH@ MOF-6 as the catalyst has been developed, which provides facile access to α …
COOH@ MOF-6 as the catalyst has been developed, which provides facile access to α …
Endogenous cell wall degrading enzyme LytD is important for the biocontrol activity of Bacillus subtilis
L Wang, J Huang, S Chen, X Su, X Zhang… - Frontiers in Plant …, 2024 - frontiersin.org
Autolysins are endogenous cell wall degrading enzymes (CWDEs) in bacteria that remodel
the peptidoglycan layer of its own cell wall. In the Bacillus subtilis genome, at least 35 …
the peptidoglycan layer of its own cell wall. In the Bacillus subtilis genome, at least 35 …
Synthesis and bioactivities of diamide derivatives containing a phenazine-1-carboxamide scaffold
X Zhu, M Zhang, L Yu, Z Xu, D Yang, X Du… - Natural product …, 2019 - Taylor & Francis
Taking natural product phenazine-1-carboxamide (PCN) as a lead compound, a series of
novel phenazine-1-carboxylic acid diamide derivatives were designed and synthesised …
novel phenazine-1-carboxylic acid diamide derivatives were designed and synthesised …
Synthesis and cytotoxic analysis of novel myrtenyl grafted pseudo-peptides revealed potential candidates for anticancer therapy
O Concepción, J Belmar, A F. de la Torre, F M. Muñiz… - Molecules, 2020 - mdpi.com
Myrtenal is a natural monoterpene isolated from essential oils of several plants and their
derivates have shown to have several biological properties including cytotoxicity. The …
derivates have shown to have several biological properties including cytotoxicity. The …
Design, synthesis and bioactivity of fluopyram derivatives containing diamide moiety
X Qingbo, L Peibo, L Huizhe, J Shuhui… - Chinese Journal of …, 2021 - sioc-journal.cn
According to the principle of combination of bioactive substructure, the structure of diamide
was introduced into fluopyram, and 22 novel fluopyram derivatives containing diamide were …
was introduced into fluopyram, and 22 novel fluopyram derivatives containing diamide were …
[HTML][HTML] 枯草芽胞杆菌基因组删减对异源酶表达影响的研究进展
张金方， 李昕悦， 徐小健， 陈雪佳， 牛馨， 任绍东… - 微生物学 …, 2021 - wswxtb.ijournals.cn
枯草芽胞杆菌作为一种遗传背景清晰, 基因编辑成熟的革兰氏阳性菌, 是多种重要工业酶的生产
宿主. 随着转录组, 蛋白质组, 代谢组等多组学测序和分析技术的发展, 通过合理设计简化枯草 …
宿主. 随着转录组, 蛋白质组, 代谢组等多组学测序和分析技术的发展, 通过合理设计简化枯草 …