Novel synthesis of quinoline chalcone derivatives-Design, synthesis, characterization and antimicrobial activity

CHP Kumar, MS Katagi, BP Nandeshwarappa - Chemical Data Collections, 2022 - Elsevier
In the present study, an easy and conventional method has been adopted for the synthesis
of novel 1-methyl-3-(3-oxo-3-phenylprop-1-enyl) quinoline-2-(1H)-ones (5a–i) by a …

Design and synthesis of novel substituted 3-(2-(1, 3, 4-thiadiazol-2-ylamino) acetyl)-2H-selenopyrano [2, 3-b] quinolin-2-ones

BP Nandeshwarappa, S Chandrashekharappa… - Chemical Data …, 2021 - Elsevier
A simple and efficient method has been developed for construction of 3-(2-(1, 3, 4-thiadiazol-
2-ylamino) acetyl)-2H-selenopyrano [2, 3-b] quinolin-2-ones (3a–f). The 3-acetyl-2H …

Selenium-Containing Heterocycles: Synthetic investigation of some new series 3-(5-mercapto-1, 3, 4-oxadiazol-2-yl)-2H-selenopyrano [2, 3-b] quinolin-2-ones

BP Nandeshwarappa, S Chandrashekharappa… - Chemical Data …, 2020 - Elsevier
Abstract A Series of hybrid 3-(5-mercapto-1, 3, 4-oxadiazol-2-yl)-2H-selenopyrano [2, 3-b]
quinolin-2-one derivatives (3a-f) were synthesized by the reaction of 2-oxo-2H …

Synthesis, characterization and structural studies of novel pyrazoline derivatives as potential inhibitors of NAD+ synthetase in bacteria and cytochrome P450 51 in …

CH Praveen Kumar, MS Katagi, J Samuel… - …, 2023 - Wiley Online Library
In the present study, a series of novel 1‐Methyl‐3‐(3‐oxo‐3‐phenylprop‐1‐enyl) quinoline‐
2‐(1H)‐ones derivatives (3 a–3 i) were synthesized via condensation, followed by the ring …

A convenient synthesis, characterization and biological evaluation of novel schiff base heterocycles as potential antimicrobial, antitubercular agents and their …

H Maruthesh, M Katagi… - Current Chemistry …, 2023 - growingscience.com
A series of (E)-1-methyl-3-((substituted phenylimino) methyl) quinolin-2 (1 H)-one schiff
bases (3a-j) bearing quinoline moiety synthesized successfully in ethanol by condensation …

Synthesis and Characterization of Substituted 5-(2-Chloroquinolin-3-yl)-1,3,4-oxadiazole-2-amines: Computational, In Silico ADME, Molecular Docking, and …

H Maruthesh, MS Katagi, J Samuel… - Russian Journal of …, 2023 - Springer
Abstract A series of 5-(2-chloroquinolin-3-yl)-1, 3, 4-oxadiazole-2-amine (IIIa–IIIj) with
different biological activities were designed and synthesized through the cyclization of …

Synthesis, computational study, solvatochromism and biological studies of thiazole-owing hydrazone derivatives

CK Yadav, BP Nandeshwarappa… - Chimica Techno …, 2023 - journals.urfu.ru
In the present work, we have synthesized thiazole-hydrazone conjugates 5 (a–h) and
characterized them using various analytical techniques such as UV, IR, NMR, and mass …

Design and Synthesis of New Series of 2-Oxo-2H-Selenopyrano[2,3-b]Quinoline-3-Carboxylates and Evaluation of Their Antibacterial Activity

S Chandrashekharappa, SO Sadashiv, SJ Patil… - Pharmaceutical …, 2022 - Springer
In the present work, newly designed ethyl 2-oxo-2 H-selenopyrano [2, 3-b] quinoline-3-
carboxylates (4a–4f) were synthesized by reaction of 3-formyl-2-selenoquinolines (3a–3f) …

Synthesis of novel pyrazolic analogues of chalcones as potential antibacterial and antifungal agents

C Kumar, S Manjunatha… - Current Chemistry …, 2023 - growingscience.com
The present includes the synthesis of pyrazoline derivatives using chalcones and phenyl
hydrazine in the presence of ethanol. It also reveals that 2-pyrazoline complexes are …

[PDF][PDF] Створення нових діуретиків на основі похідних хінолону-2

МЮ Голік - 2021 - dspace.nuph.edu.ua
Національний фармацевтичний університет Міністерство охорони здоро Page 1
Національний фармацевтичний університет Міністерство охорони здоров’я України …