Recent Progress in the Synthesis and Biological Assessment of Benzimidazole-1, 2, 3-Triazole Hybrids

DK Singh, H Iqbal, MA Ansari - Current Organic Chemistry, 2024 - benthamdirect.com
In recent times, many research groups have focused their attention on nitrogencontaining
heterocyclic compounds with the aim of gaining a deeper understanding of their biological …

[HTML][HTML] Antibacterial Activity and Antifungal Activity of Monomeric Alkaloids

AM Thawabteh, AW Ghanem, S AbuMadi, D Thaher… - Toxins, 2024 - mdpi.com
Scientists are becoming alarmed by the rise in drug-resistant bacterial and fungal strains,
which makes it more costly, time-consuming, and difficult to create new antimicrobials from …

Synthesis anticancer evaluation and molecular docking studies of Amide derivatives of Oxazole-Pyrimidine-1, 3, 4-Thiadiazole analogues

MR Veeraboina, V Pattabi, N Somaiah… - Chemical Data …, 2023 - Elsevier
A new library of amide derivatives of oxazole-pyrimidine-1, 3, 4-thiadiazoles (11a-j) was
conceived and developed, with their chemical structures validated by 1 HNMR, 13 CNMR …

New Dipterocarpol‐Based Molecules with α‐Glucosidase Inhibitory and Hypoglycemic Activity

IE Smirnova, ZI Galimova, TA Sapozhnikova… - …, 2024 - Wiley Online Library
Dammarane triterpenoids are affordable and bioactive natural metabolites with great
structural potential, which makes them attractive sources for drug development. The aim of …

Lewis acid-mediated transformations of 5-acyl-N-fluoroalkyl-1, 2, 3-triazoles to cyclopentenones, indenones, or oxazoles

L Janecký, P Beier - RSC advances, 2024 - pubs.rsc.org
We present a transition metal-free approach to 2-N-substituted indenones, cyclopentenones,
and 4-carbonyl oxazoles, based on the reaction of 5-acylated N-fluoroalkyl substituted 1, 2 …

[HTML][HTML] Non-nucleophilic base promoted synthesis of azo-linked oxazolone-pyrazole hybrids: Antimicrobial, antitubercular, anticancer evaluations and in-silico …

BY Patel, V Joshi, S Subramanian, G Italiya… - Results in …, 2024 - Elsevier
Ten new non-nucleophilic base (DBU) catalyzed oxazolone-bearing pyrazole derivatives
were created to treat infectious diseases caused by bacterial, mycobacterial strains, and …

Electrochemical Determination of Cysteine Using a 2-(2, 5-Dihydroxy-Phenyl)-Naphtho [1, 2-d] Oxazole-5-Sulfonic Acid (DHPNOS) and Cerium Oxide Nanoparticle …

L Darboe, A Benvidi, E Amin Sadrabadi… - Analytical …, 2024 - Taylor & Francis
An electrochemical sensor for the electrocatalytic oxidation of cysteine was designed based
upon a 2-(2, 5-dihydroxy-phenyl)-naphtho [1, 2-d] oxazole-5-sulfonic acid (DHPNOS) and …

Hybrids of Benzimidazole-oxadiazole: A New Avenue for Synthesis, Pharmacological Activity and Recent Patents for the Development of More Effective Ligands

G Bhasker, Salahuddin, A Mazumder… - Current Organic …, 2024 - benthamdirect.com
Background: Two significant families of compounds ie 1, 3, 4-oxadiazole and
benzimidazole, have undergone extensive investigation into their pharmacological …

Phosphorus-Containing Alkynes in the Synthesis of Heterocyclic Compounds (A Review)

AA Sokolov, DM Egorov, AV Dogadina… - Russian Journal of …, 2024 - Springer
Phosphorus-substituted heterocycles are an important class of organophosphorus
compounds that are widely used in the drug development, agrochemistry, materials science …

Cerric ammonium nitrate catalyzed eco-friendly green synthesis of chitosan Schiff base using PEG-400 as an anticancer agent against gastric cancer cells via …

W Geng, X Feng, C Li, S Ni - Bulletin of the Chemical Society of Ethiopia, 2024 - ajol.info
The present study was conducted to scrutinize the pharmacological effect of oxazole-
embedded Chitosan as an anticancer agent against gastric cancer cells. This compound …