[PDF][PDF] Synthesis and Biological Evaluation of Five-and Six-Membered Heterocycles as an Anti-Diabetic Agent: An Overview

GP Sadawarte, JD Rajput, AD Kale, VB Jagrut - Journal of Chemical Reviews, 2024 - sid.ir
Archive of SID.ir Archive of SID.ir Page 1 2024, Volume 6, Issue 3 331 Journal of Chemical
Reviews *Corresponding Author: Gautam P. Sadawarte (gautamsadawarte@gmail.com ) …

Synthesis and tyrosinase inhibitory activities of 4-oxobutanoate derivatives of carvacrol and thymol

N Brotzman, Y Xu, A Graybill, A Cocolas… - Bioorganic & medicinal …, 2019 - Elsevier
Abstract Carvacrol (1) and thymol (2) were converted to their alkyl 4-oxobutanoate
derivatives (7–20) in three steps, and evaluated for tyrosinase inhibitory activity. The …

Synthesis, characterizations, biological activities and docking studies of novel dihydroxy derivatives of natural phenolic monoterpenoids containing azomethine …

JD Rajput, SD Bagul, AA Hosamani, MM Patil… - Research on Chemical …, 2017 - Springer
In the present work, we report the synthesis of six new azomethine linkage containing
dihydroxy derivatives of carvacrol, thymol, and eugenol. All the synthesized derivatives have …

Microwave-promoted synthesis of highly luminescent s-tetrazine-1, 3, 4-oxadiazole and s-tetrazine-1, 3, 4-thiadiazole hybrids

A Kędzia, A Kudelko, M Świątkowski, R Kruszyński - Dyes and Pigments, 2020 - Elsevier
Two series of new s-tetrazine derivatives containing 1, 3, 4-oxadiazole and 1, 3, 4-
thiadiazole rings were synthesized from s-tetrazine-3, 6-dicarbohydrazide, triethyl …

Antioxidant and tyrosinase docking studies of heterocyclic sulfide derivatives containing a thymol moiety

MH Havasi, AJ Ressler, EL Parks, AH Cocolas… - Inorganica Chimica …, 2020 - Elsevier
Abstract Fourteen heterocyclic sulfide derivatives (4–17) containing a thymol moiety and
oxadiazole, thiadiazole, triazole, oxazole, thiazole, imidazole, pyridine or purine …

Synthesis, biological activities and molecular docking simulation of hydrazone scaffolds of carvacrol, thymol and eugenol

JD Rajput, SD Bagul, RS Bendre - Research on Chemical Intermediates, 2017 - Springer
In present work, we report the synthesis of 12 new hydrazones and sulfonyl hydrazones
linkage containing carvacrol, thymol and eugenol derivatives by simple condensation …

2-isopropyl-4-methoxy-5-methylphenol-hydrazone derivatives: Synthesis, characterization, and in-silico assessment of EGFR and Bcl2 inhibitory activity

Y Laamari, AN Ousidi, A Bimoussa, MT Rehman… - Journal of Molecular …, 2025 - Elsevier
The exploration of hydrazones, characterized by the-N (H) N= CH group, in combination with
thymol, has garnered significant attention in pharmacology due to their versatility and ease …

[图书][B] Terpenoids: Chemistry, Biochemistry, Medicinal Effects, Ethno-pharmacology

BK Banik, BM Sahoo, A Tiwari - 2022 - taylorfrancis.com
This unique volume covers specific aspects of the biological chemistry of terpenoids. It
provides extensive information related to classification, general methods of extraction and …

Synthesis, characterization, and antioxidant activity of thymol-based paracetamol analogues

PS Sathe, JD Rajput, SS Gunaga, HM Patel… - Research on chemical …, 2019 - Springer
Abstract Thymol (2-isopropyl-5-methylphenol) is an important monoterpene phenol
occurring in the essential oils isolated from Thymus vulgaris, Thymus zygis, Thymus …

Insect growth regulatory activity of carvacrol-based 1, 3, 4-thiadiazoles and 1, 3, 4-oxadiazoles

SD Bagul, JD Rajput, C Srivastava, RS Bendre - Molecular Diversity, 2018 - Springer
Abstract In designing of novel insect growth regulators (IGRs), biologically occurring
carvacrol has been structurally modified to thiadiazole and oxadiazole moieties. Two series …