Potassium Poly (Heptazine Imide): Transition Metal‐Free Solid‐State Triplet Sensitizer in Cascade Energy Transfer and [3+ 2]‐cycloadditions

A Savateev, NV Tarakina, V Strauss… - Angewandte Chemie …, 2020 - Wiley Online Library
Polymeric carbon nitride materials have been used in numerous light‐to‐energy conversion
applications ranging from photocatalysis to optoelectronics. For a new application and …

Investigating the Influence of (Deoxy)fluorination on the Lipophilicity of Non‐UV‐Active Fluorinated Alkanols and Carbohydrates by a New log P Determination …

B Linclau, Z Wang, G Compain… - Angewandte Chemie …, 2016 - Wiley Online Library
Property tuning by fluorination is very effective for a number of purposes, and currently
increasingly investigated for aliphatic compounds. An important application is lipophilicity …

Advancing the drug discovery and development process

KC Nicolaou - Angewandte Chemie, 2014 - Wiley Online Library
The current state of affairs in the drug discovery and development process is briefly
summarized and then ways to take advantage of the ever‐increasing fundamental …

General α‐amino 1, 3, 4‐oxadiazole synthesis via late‐stage reductive functionalization of tertiary amides and lactams

D Matheau‐Raven, DJ Dixon - … Chemie International Edition, 2021 - Wiley Online Library
An iridium‐catalyzed reductive three‐component coupling reaction for the synthesis of
medicinally relevant α‐amino 1, 3, 4‐oxadiazoles from abundant tertiary amides or lactams …

Batch versus flow lithiation–substitution of 1, 3, 4‐oxadiazoles: Exploitation of unstable intermediates using flow chemistry

JYF Wong, JM Tobin, F Vilela… - Chemistry–A European …, 2019 - Wiley Online Library
Oxadiazoles are a common motif in pharmaceutical chemistry, but few convenient methods
for their modification exist. A fast, convenient, high yielding and general α‐substitution of 1 …

1, 2, 4‐and 1, 3, 4‐Oxadiazole synthesis by palladium‐catalyzed carbonylative assembly of aryl bromides with amidoximes or hydrazides

TL Andersen, W Caneschi, A Ayoub… - Advanced Synthesis …, 2014 - Wiley Online Library
Aryl bromides were successfully transformed into their corresponding N, N′‐
diacylhydrazines via a Pd‐catalyzed carbonylative coupling with acylhydrazines. These …

A metal-free tandem approach to prepare structurally diverse N-heterocycles: synthesis of 1, 2, 4-oxadiazoles and pyrimidinones

PK Gupta, MK Hussain, M Asad, R Kant… - New Journal of …, 2014 - pubs.rsc.org
A metal-free one-pot approach to the diversity oriented synthesis of N-heterocycles, 1, 2, 4-
oxadiazoles and 2, 6 disubstituted pyrimidin-4-ones is described via carboxamidation of …

Synthesis of novel indole‐oxadiazole molecular hybrids by a regioselective C‐3 sulfenylation of indole with 1, 3, 4‐oxadiazole‐2‐thiols using iodine‐dimethyl …

K Dutta, AG Majumdar, N Kushwah… - Journal of …, 2022 - Wiley Online Library
Novel indole‐oxadiazole molecular hybrids have been synthesized by a regioselective C‐3
sulfenylation of indoles with 1, 3, 4‐oxadiazole‐2‐thiols for the first time using iodine as a …

UV‐induced 1, 3, 4‐oxadiazole formation from 5‐substituted tetrazoles and carboxylic acids in flow

L Green, K Livingstone, S Bertrand… - … A European Journal, 2020 - Wiley Online Library
Abstract A range of 1, 3, 4‐oxadiazoles have been synthesized using a UV‐B activated flow
approach starting from carboxylic acids and 5‐substituted tetrazoles. The application of UV …

Green Synthetic Approach for the Construction of 3, 5‐Disubstituted 1, 2, 4‐Oxadiazoles and Ataluren Analogues from Dithioesters Using Water

HA Swarup, N Chaithra, K Mantelingu… - …, 2018 - Wiley Online Library
An innovative green synthesis of 3, 5‐disubstituted 1, 2, 4‐oxadiazoles from dithioesters
using water as a solvent. This approach becomes more interesting because it undergoes …