Natural product synthesis is a highly demanding field in constant need of efficient
transformations that allow either straightforward, scalable, and high-yielding preparation of …

Transition metal-catalyzed cross-coupling reactions of alkyl metals and aryl halides or
pseudohalides have emerged as a powerful methodology for the formation of Csp3-Csp2 …

Substituted heterocycles are a structural component of a vast number of biologically active
natural and non-natural compounds. Synthesis of various heterocycles has been a research …

The indole unit is one of the most abundant and relevant heterocycles in natural products
and pharmaceuticals.[1] Despite the existence of numerous methods for the synthesis and …

Providing comprehensive insight into the use of copper in cross-coupling reactions, Copper-
Mediated Cross-Coupling Reactions provides a complete up-to-date collection of the …

Abstract The direct C H annulation of anilines or related compounds with internal alkynes
provides straightforward access to 2, 3‐disubstituted indole products. However, this …

The synthesis of N-heterocyclic compounds is an important direction because of their
diverse biological functions. Recently, there has been remarkable progress in copper …

A concise approach to various benzisothiazol-3 (2 H)-one derivatives has been developed
by copper-catalyzed the reaction of o-bromobenzamide derivatives with potassium …

Copper-catalyzed domino reactions are one of the most useful strategies for the construction
of various cyclic compounds. In this Synopsis, we mainly focus on the latest advances in …

Multisubstituted indoles were synthesized via a one-pot tandem copper-catalyzed Ullmann-
type C–N bond formation/intramolecular cross-dehydrogenative coupling process at 130° C …