[PDF][PDF] Pyrazoline derivatives: a worthy insight into the recent advances and potential pharmacological activities

MA Rahman, AA Siddiqui - Int J Pharm Sci Drug Res, 2010 - researchgate.net
Pyrazolines display a broad spectrum of potential pharmacological activities and are present
in a number of pharmacologically active molecules such as phenazone/amidopyrene …

Biological activities of pyrazoline derivatives-A recent development

S Kumar, S Bawa, S Drabu, R Kumar… - Recent patents on anti …, 2009 - ingentaconnect.com
Pyrazolines are well known and important nitrogen containing 5-membered heterocyclic
compounds and various methods have been worked out for their synthesis. Numerous …

[HTML][HTML] Synthesis, antibacterial and antifungal activity of some new pyrazoline and pyrazole derivatives

SY Hassan - Molecules, 2013 - mdpi.com
A series of 2-pyrazolines 5–9 have been synthesized from α, β-unsaturated ketones 2–4.
New 2-pyrazoline derivatives 13–15 bearing benzenesulfonamide moieties were then …

Recent advances in the therapeutic applications of pyrazolines

MR Shaaban, AS Mayhoub… - Expert opinion on …, 2012 - Taylor & Francis
Introduction: Pyrazolines are well-known and important nitrogen-containing five-membered
ring heterocyclic compounds. Various methods have been worked out for their synthesis …

Pyrazolines: a biological review

A Marella, R Ali, T Alam, R Saha… - Mini reviews in …, 2013 - ingentaconnect.com
Pyrazoline is an important five membered nitrogen heterocycle, which has been extensively
researched upon. The ring is quite stable and has inspired chemists to carry out various …

Epidermal growth factor receptor inhibitors as potential anticancer agents: An update of recent progress

B Sharma, VJ Singh, PA Chawla - Bioorganic Chemistry, 2021 - Elsevier
Epidermal growth factor receptor (EGFR) is a vital intermediate in cell signaling pathway
including cell proliferation, angiogenesis, apoptosis, and metastatic spread and also having …

Synthesis of some new 2-(3-pyridyl)-4, 5-disubstituted thiazoles as potent antimicrobial agents

S Bondock, T Naser, YA Ammar - European Journal of Medicinal Chemistry, 2013 - Elsevier
As a part of ongoing studies in developing new potent antimicrobial agents, a series of novel
2-(3-pyridyl)-4, 5-disubstituted thiazoles was efficiently synthesized and characterized by …

[HTML][HTML] Synthesis, antimicrobial and antitubercular activities of some novel pyrazoline derivatives

A Ahmad, A Husain, SA Khan, M Mujeeb… - Journal of Saudi …, 2016 - Elsevier
In the present study, two new series of pyrazolines (3a–h & 4a–h) were synthesized starting
from p-acetamidophenol (paracetamol) and evaluated for their antibacterial, antifungal and …

[HTML][HTML] Synthesis and anticonvulsant activity of some 2-pyrazolines derived from chalcones

N Beyhan, B Kocyigit-Kaymakcioglu, S Gümrü… - Arabian Journal of …, 2017 - Elsevier
Abstract Synthesis of chalcones (1, 3-diarylprop-2-en-1-ones) and 2-pyrazoline derivatives
has been an active field of research due to their established pharmacological effects. In this …

Synthesis, QSAR and anticandidal evaluation of 1, 2, 3-triazoles derived from naturally bioactive scaffolds

M Irfan, B Aneja, U Yadava, SI Khan, N Manzoor… - European Journal of …, 2015 - Elsevier
In the present study, we used eight natural precursors (1a-h) with most of them having
promising antimicrobial activities and synthesised their novel 1, 2, 3-triazole derivatives (3a …