Evaluation of synthetic 2-aryl quinoxaline derivatives as α-amylase, α-glucosidase, acetylcholinesterase, and butyrylcholinesterase inhibitors
Variety of 2-aryl quinoxaline derivatives 1–23 were synthesized in good yields, by reacting
1, 2-phenylenediamine with varyingly substituted phenacyl bromides in the presence of …
1, 2-phenylenediamine with varyingly substituted phenacyl bromides in the presence of …
Fluorinated benzimidazolium salts: Synthesis, characterization, molecular docking studies and inhibitory properties against some metabolic enzymes
Here, a number of symmetric and unsymmetric N-heterocyclic carbene (NHC) precursors
based on benzimidazol-2-ylidene are synthesized. The N-benzyl substituent in these …
based on benzimidazol-2-ylidene are synthesized. The N-benzyl substituent in these …
Sc3+ Chloro and Alkyl Complexes Coordinated by Pincer NHC‐Tethered Bis(phenolate) Ligands
GA Gurina, AV Markin, AV Cherkasov… - European Journal of …, 2023 - Wiley Online Library
Bis (phenolate) ligands with benzimidazole‐2‐ylidene (L1) and tetrahydropyrimidine‐2‐
ylidene (L2) linkers proved to be suitable coordination environments for the synthesis of …
ylidene (L2) linkers proved to be suitable coordination environments for the synthesis of …
Benzimidazolium Salts Containing Trifluoromethoxybenzyl: Synthesis, Characterization, Crystal Structure, Molecular Docking Studies and Enzymes Inhibitory …
The method for producing 4‐trifluoromethoxybenzyl substituted benzimidazolium salts is
described in this article. The method is based on the reaction of 4‐trifluoromethoxybenzyl …
described in this article. The method is based on the reaction of 4‐trifluoromethoxybenzyl …
Acetylphenyl-substituted imidazolium salts: synthesis, characterization, in silico studies and inhibitory properties against some metabolic enzymes
Herein, we present how to synthesize thirteen new 1-(4-acetylphenyl)-3-alkylimidazolium
salts by reacting 4-(1-H-imidazol-1-yl) acetophenone with a variety of benzyl halides that …
salts by reacting 4-(1-H-imidazol-1-yl) acetophenone with a variety of benzyl halides that …
Design, synthesis, spectroscopic characterizations, single crystal X-ray analysis, in vitro xanthine oxidase and acetylcholinesterase inhibitory evaluation as well as in silico …
Herein, eight new NHC-based selenourea derivatives were synthesized and characterized
by using spectroscopic method (1H, 19F, and 13C NMR, FT-IR), and elemental analysis …
by using spectroscopic method (1H, 19F, and 13C NMR, FT-IR), and elemental analysis …
Thioether-substituted Benzimidazolium Salts: Synthesis, Characterization, Crystal Structure, and Their Inhibitory Properties Against Acetylcholinesterase and Xanthine …
The sulfurous compounds are known as organosulfur, which has been associated with
numerous biological activities in both natural products and synthetic organic compounds. In …
numerous biological activities in both natural products and synthetic organic compounds. In …
[HTML][HTML] Impact of Synthesized Zero-valance Silver Nanoparticles on Acetylcholinesterase and Xanthine Oxidase: Toxicological and Environmental Implications
SH Mohammed, AM Rheima, DA Al-aameri… - Case Studies in …, 2025 - Elsevier
Nanoparticles have several applications in commercial and pharmaceutical products owing
to their exceptional antibacterial characteristics. Nonetheless, the extensive creation of …
to their exceptional antibacterial characteristics. Nonetheless, the extensive creation of …
Synthesis, characterization and inhibitor properties of benzimidazolium salts bearing 4-(methylsulfonyl) benzyl side arms
Herein, a series of N-heterocyclic carbene (NHC) precursors bearing sulfonyl moieties was
prepared. 1-(4-(methylsulfonyl) benzyl)-3-alkylbenzimidazolium chloride salts were …
prepared. 1-(4-(methylsulfonyl) benzyl)-3-alkylbenzimidazolium chloride salts were …
Benzimidazolium Salts Bearing Nitrile Moieties: Synthesis, Enzyme Inhibition Profiling, and Molecular Docking Analysis for Carbonic Anhydrase and …
This report presents the synthesis and characterization of a range of benzimidazolium salts
featuring 3‐cyanopropyl groups on the 1st nitrogen atom and varied alkyl groups on the 3rd …
featuring 3‐cyanopropyl groups on the 1st nitrogen atom and varied alkyl groups on the 3rd …