The indole alkaloids, ranging from lysergic acid to vincristine, have long inspired organic
synthesis chemists. Interest in developing new methods for indole synthesis has burgeoned …

Despite the importance in synthetic, agrochemical, and medicinal chemistry, to the best of
our knowledge, no overview has been made on the synthetic methods and the field of …

The palladium-catalyzed coupling of 2-iodoaniline and the corresponding N-methyl,-acetyl,
and-tosyl derivatives with a wide variety of internal alkynes provides 2, 3-disubstituted …

Zn (OTf) 2 (10 mol%) catalyzed the cyclization of propargyl alcohols with PhXH (X= O, NH) in
hot toluene (100 οC) without additive and gave indole and benzofuran products with …

One-pot synthesis of indoles by a palladium-catalyzed annulation of ortho-haloanilines and
aldehydes has been developed. Coupling of ortho-iodoaniline with aldehyde is realized …

A variety of substituted enamine derivatives were first found to be conveniently converted to
the corresponding 2 H-azirines mediated by phenyliodine (III) diacetate (PIDA). The formed …

Two complementary procedures have been developed for the conversion of the oximes of α-
aryl ketones to azirines. On heating, the azirines rearrange smoothly to the corresponding …

An efficient and stereoselective synthesis of vinylphosphonates and phosphine oxides was
developed starting from styrenes using AgNO3 as the catalyst and K2S2O8 as the oxidant …

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The word indole is derived from the word India: indigo (3), the blue dye, was first exported
from India to Europe in the 16th century. Indoles are generally crystalline colorless solids …