Versatile Therapeutic Values of N‐Containing Heterocycles Benzimidazole, Piperazine and Piperidine Hybrids

AR Zala, P Kumari - ChemistrySelect, 2023 - Wiley Online Library
Nitrogen‐containing benzimidazole, piperazine, and piperidine are significant
pharmacophores in medicinal chemistry and drug development. Many medications, lead …

Computational and Experimental Investigation of Antibacterial Properties of Some Fluorinated Thioureas

AA Tagiling, WM Khairul, R Rahamathullah… - Polycyclic Aromatic …, 2023 - Taylor & Francis
Herein, fluorinated thioureas with various substituents (F1-F3) were synthesized and
characterized spectroscopically and analytically to investigate their properties as …

Multiple molecular targets mediated antioxidant activity, molecular docking, ADMET, QSAR and bioactivity studies of halo substituted urea derivatives of α-Methyl-l …

N Vadabingi, VKR Avula, GV Zyryanov, S Vallela… - Bioorganic …, 2020 - Elsevier
A series of novel α-methyl-l-DOPA urea derivatives viz., 3-(3, 4-dihydroxyphenyl)-2-methyl-2-
(3-halo/trifluoromethyl substituted phenyl ureido) propanoic acids (6a-e) have been …

[HTML][HTML] Evaluation of a new benzothiazole derivative with antioxidant activity in the initial phase of acetaminophen toxicity

LC Cabrera-Perez, II Padilla-Martínez, A Cruz… - Arabian Journal of …, 2019 - Elsevier
Increasing evidence indicates that benzothiazoles and thioureas have the ability to
inactivate reactive chemical species through their antioxidant activity. In this context, we …

Synthesis and characterization of new fluoro/trifluoromethyl-substituted acylthiourea derivatives with promising activity against planktonic and biofilm-embedded …

C Limban, DC Nuta, AV Missir, R Roman, MT Caproiu… - Processes, 2020 - mdpi.com
The aim of this study was preparation of new derivatives based on 2-((4-chlorophenoxy)
methyl)-N-(arylcarbamothioyl) benzamide structure; the new compounds were characterized …

Palladium-coated thiourea core-shell nanocomposite as a new, efficient, and magnetic responsive nanocatalyst for the Suzuki-Miyaura coupling reactions

R Eivazzadeh-Keihan, N Bahrami… - Materials Research …, 2021 - iopscience.iop.org
In this research, according to the important aspects of palladium components in conducting
Suzuki-Miyaura coupling reactions and formation of biphenyl compounds, magnetic …

Design, synthesis, in vitro and in silico bioactivity profiles of new urea/thiourea derivatives of 2-pyridyl piperazine as potent antioxidant and antimicrobial agents …

S Sumalatha, C Venkataramaiah… - Journal of Biomolecular …, 2023 - Taylor & Francis
Synthesis of a series of new urea and thiourea derivatives of 2-pyridyl piperazine was
accomplished by reacting various isocyanates and isothiocyanates in the presence of …

In silico and in vitro antioxidant and anticancer activity profiles of urea and thiourea derivatives of 2,3-dihydro-1H-inden-1-amine

M Chandrasekhar, G Syam Prasad… - Journal of Receptors …, 2020 - Taylor & Francis
Synthesis of a series of new urea and thiourea compounds have been accomplished by the
reaction of 2, 3-dihydro-1 H-inden-1-amine with various phenyl isocyanates and …

Design and Straightforward Synthesis of Novel N-substituted 6-Fluoro-3-(piperidin-4-yl)-1, 2-benzoxazole Derivatives and Their Antibacterial Activity

KK Garlapati, RK Ganta, KS Kumar… - Russian Journal of …, 2023 - Springer
A facile synthetic route to N-substituted 6-fluoro-3-(piperidin-4-yl)-1, 2-benzoxazole
derivatives using piperidine-4-carboxylic acid, 1, 3-difluorobenzene, and various halogen …

[PDF][PDF] Synthesis of Some New Chrysin Derivatives and Their Biological Assessment as Antibacterial, Antibiofilm and Antifungal Agent.

S Bhowmik, T Das, S Ghosh, BK Sharma… - Asian Journal of …, 2018 - academia.edu
Some new derivatives of natural chrysin have been synthesized and evaluated for
antibacterial, antibiofilm and antifungal activities. Three compounds, namely 2a, 2e, 2i …