Synthesis, antimicrobial activities, docking studies and computational calculations of new bis-1,4-phenylene -1H-1,2,3-triazole derivatives utilized ultrasonic energy
S Soror, AM Fahim, S Elabbady, E Nassar… - Journal of …, 2022 - Taylor & Francis
In this elucidation, we studied the utility of condensation reaction between 1, 4-
phenylenediamine (1) with acetyl acetone (2) with hydrazine hydrate utilized ultrasonic …
phenylenediamine (1) with acetyl acetone (2) with hydrazine hydrate utilized ultrasonic …
Design, synthesis, spectroscopic characterization, in-vitro antibacterial evaluation and in-silico analysis of polycaprolactone containing chitosan-quercetin …
Aim of present study was to synthesize a novel chitosan-quercetin (CTS-QT) complex by
making a carbodiimide linkage using maleic anhydride as cross-linker and to investigate its …
making a carbodiimide linkage using maleic anhydride as cross-linker and to investigate its …
Design, synthesis, in vitro anti-oxidant evaluation, α-amylase inhibition assay, and molecular docking analysis of 2-(2-benzylidenehydrazinyl)-4, 4-diphenyl-1H …
Reactive oxygen and nitrogen species (RONS) regulate physiological processes to ensure
cellular integrity. However, overproduction of RONS leads to oxidative stresses which results …
cellular integrity. However, overproduction of RONS leads to oxidative stresses which results …
The development of novel cytochrome P450 2J2 (CYP2J2) inhibitor and the underlying interaction between inhibitor and CYP2J2
X Tian, M Zhou, J Ning, X Deng, L Feng… - Journal of Enzyme …, 2021 - Taylor & Francis
Abstract Human Cytochrome P450 2J2 (CYP2J2) as an important metabolic enzyme, plays
a crucial role in metabolism of polyunsaturated fatty acids (PUFAs). Elevated levels of …
a crucial role in metabolism of polyunsaturated fatty acids (PUFAs). Elevated levels of …
Exploring Acyl Thiotriazinoindole Based Pharmacophores: Design, Synthesis, and SAR Studies with Molecular Docking and Biological Activity Profiling against Urease, α …
A diminutive chemical library of acyl thiotriazinoindole (ATTI) based bioactive scaffolds was
synthesized, instigated by taking the economical starting material Isatin, through a series of …
synthesized, instigated by taking the economical starting material Isatin, through a series of …
Synthesis, in silico guided DNA-interaction analysis, in vitro anti-oxidant evaluation, and antibacterial assay of 4-amino-5-(2-benzylidenehydrazinyl)-2 H-1, 2, 4 …
The current research contains synthesis, DNA-interaction analysis, in vitro anti-oxidant
evaluation, and antibacterial assay of triazole-azomethine hybrids. Consequently, the …
evaluation, and antibacterial assay of triazole-azomethine hybrids. Consequently, the …
Evaluation of Ternary Thiazole-Coumarin-Azomethine Derivatives as Multi-Target Inhibitors: α-Amylase, Urease, Free Radical Scavenging and Antibacterial Activities …
Present studies primarily demonstrate the evaluation of ternary thiazole-coumarin-
azomethine derivatives for their in-vitro assessment against α-amylase, urease …
azomethine derivatives for their in-vitro assessment against α-amylase, urease …
Design, synthesis, and antiproliferative investigation of novel quinazolinones incorporating 1, 3, 4-oxadiazole and 1, 2, 4-triazole thioether moieties
Z Li, Y Men, S Gao, P Cui, H Wang… - Phosphorus, Sulfur, and …, 2024 - Taylor & Francis
In the current study, a series of 1, 3, 4-oxadiazole and 1, 2, 4-triazole derivatives linked to
quinazolinone were designed and synthesized by using Phase Transfer Catalysis. The …
quinazolinone were designed and synthesized by using Phase Transfer Catalysis. The …