Thiazole-containing compounds as therapeutic targets for cancer therapy
In the last few decades, considerable progress has been made in anticancer agents
development, and several new anticancer agents of natural and synthetic origin have been …
development, and several new anticancer agents of natural and synthetic origin have been …
Visible light photocatalysis in the synthesis of pharmaceutically relevant heterocyclic scaffolds
Visible light and photoredox catalysis have emerged as a powerful and long-lasting tool for
organic synthesis, demonstrating the importance of a variety of chemical bond formation …
organic synthesis, demonstrating the importance of a variety of chemical bond formation …
Bioactive thiazole and benzothiazole derivatives
The heterocycles are the versatile compounds existing in almost all natural products and
synthetic organic compounds, usually associated with one or the other biological activity …
synthetic organic compounds, usually associated with one or the other biological activity …
Thiazole in the targeted anticancer drug discovery
A Ayati, S Emami, S Moghimi… - Future medicinal …, 2019 - Taylor & Francis
Cancer is known as one of the main causes of death in the world; and many compounds
have been synthesized to date with potential use in cancer therapy. Thiazole is a versatile …
have been synthesized to date with potential use in cancer therapy. Thiazole is a versatile …
Design, synthesis and docking studies of novel thiazole derivatives incorporating pyridine moiety and assessment as antimicrobial agents
RE Khidre, IAM Radini - Scientific reports, 2021 - nature.com
A novel series of substituted 4, 6-dimethyl-2-oxo-1-(thiazol-2-ylamino)-1, 2-dihydropyridine-
3-carbonitrile derivatives 6, 9, 13, 15, and 17 was synthesized in a good to excellent yield …
3-carbonitrile derivatives 6, 9, 13, 15, and 17 was synthesized in a good to excellent yield …
Design, synthesis and molecular docking of new pyrazole-thiazolidinones as potent anti-inflammatory and analgesic agents with TNF-α inhibitory activity
SS Abd El-Karim, HS Mohamed, MF Abdelhameed… - Bioorganic …, 2021 - Elsevier
A new set of derivatives bearing pyrazole-methylenehydrazono-thiazolidinone scaffold 4–23
was designed, synthesized and confirmed by different spectroscopic means and elemental …
was designed, synthesized and confirmed by different spectroscopic means and elemental …
Thiazoles: having diverse biological activities
In the last few decades, a lot of work has been done on thiazole ring to find new compounds
related to this scaffold to act as antioxidant, analgesic, anti-inflammatory, antimicrobial …
related to this scaffold to act as antioxidant, analgesic, anti-inflammatory, antimicrobial …
Antimicrobial and antioxidant activities of Streptomyces species from soils of three different cold sites in the Fez-Meknes region Morocco
S Rammali, L Hilali, K Dari, B Bencharki, A Rahim… - Scientific reports, 2022 - nature.com
The increasing demand for new bioactive compounds to combat the evolution of multi-drug
resistance (MDR) requires research on microorganisms in different environments in order to …
resistance (MDR) requires research on microorganisms in different environments in order to …
Novel class of benzimidazole-thiazole hybrids: The privileged scaffolds of potent anti-inflammatory activity with dual inhibition of cyclooxygenase and 15-lipoxygenase …
MTE Maghraby, OMF Abou-Ghadir… - Bioorganic & medicinal …, 2020 - Elsevier
The present study includes design and synthesis of new molecular hybrids of 2-
methylthiobenzimidazole linked to various anti-inflammatory pharmacophores through 2 …
methylthiobenzimidazole linked to various anti-inflammatory pharmacophores through 2 …
[PDF][PDF] Thiazoles: a valuable insight into the recent advances and biological activities
Thiazoles displayed broad range of biological activities and found in many potent
biologically active molecules such as Sulfathiazol (antimicrobial drug), Ritonavir …
biologically active molecules such as Sulfathiazol (antimicrobial drug), Ritonavir …