The late stage functionalization (LSF) of complex biorelevant compounds is a powerful tool
to speed up the identification of structure–activity relationships (SARs) and to optimize …

Over the past few decades, the advent of C–H activation has led to a rethink among
chemists about the synthetic strategies employed for multi-step transformations. Indeed …

Azines, which are six-membered aromatic compounds containing one or more nitrogen
atoms, serve as ubiquitous structural cores of aromatic species with important applications in …

The direct functionalization of C H bonds in organic compounds has recently emerged as a
powerful and ideal method for the formation of carbon–carbon and carbon–heteroatom …

In recent years, transition metal‐catalyzed direct (hetero) arylation reactions of heteroarenes
with (hetero) aryl halides and pseudohalides have received significant attention as eco …

Die direkte Funktionalisierung von C‐H‐Bindungen in organischen Molekülen hat sich in
jüngster Zeit zu einer wirksamen und idealen Methode entwickelt, mit der Kohlenstoff …

We report herein the iridium-catalyzed meta-selective C–H borylation of benzamides by
using a newly designed 2, 2′-bipyridine (bpy) ligand bearing an alkylaluminum …

Quinoline is an important scaffold in many natural products, biologically active compounds,
and functional materials. The C–H functionalization of quinoline scaffolds by transition metal …

Methods that directly functionalize pyridines are in high demand due to their presence in
pharmaceuticals, agrochemicals, and materials. A reaction that selectively transforms the 4 …

Pyridines and related N-heteroarenes are commonly found in pharmaceuticals,
agrochemicals and other biologically active compounds,. Site-selective C–H …