Comprehensive Coverage on Anti‐mycobacterial Endeavour Reported in 2021
TM Dhameliya, AA Devani, KA Patel… - ChemistrySelect, 2022 - Wiley Online Library
Tuberculosis (TB) has been the highly contagious airborne disease caused by
Mycobacterium tuberculosis and the major leading infectious disease with the higher …
Mycobacterium tuberculosis and the major leading infectious disease with the higher …
Design, Synthesis, Molecular docking, and biological evaluation of novel 2, 3-diaryl-1, 3-thiazolidine-4-one derivatives as potential anti-inflammatory and cytotoxic …
YO Mekhlef, AM AboulMagd, AM Gouda - Bioorganic Chemistry, 2023 - Elsevier
Abstract A new series of 2, 3-diaryl-1, 3thiazolidin-4-one derivatives was designed,
synthesized, and evaluated for their cytotoxicity and COXs inhibitory activities. Among these …
synthesized, and evaluated for their cytotoxicity and COXs inhibitory activities. Among these …
Synthesis, SC-XRD structure, spectroscopy, intermolecular interactions, DFT/TD-DFT investigation, and (static, dynamic) NLO properties of (2E, 5Z)-3-(4-fluorophenyl) …
N Kheddam, A Djafri, Y Megrouss, R Rahmani… - Journal of Molecular …, 2024 - Elsevier
This paper describes the synthesis of a novel fluorine-substituted thiazolidin-4-one
compound,(2E, 5Z)-3-(4-fluorophenyl)-2-(4-fluorophenylimino)-5-((E)-3-(2-nitrophenyl) …
compound,(2E, 5Z)-3-(4-fluorophenyl)-2-(4-fluorophenylimino)-5-((E)-3-(2-nitrophenyl) …
[HTML][HTML] Discovery of two non-UDP-mimic inhibitors of O-GlcNAc transferase by screening a DNA-encoded library
C Balsollier, S Bijkerk, A de Smit, K van Eekelen… - Bioorganic …, 2024 - Elsevier
Finding potent inhibitors of O-GlcNAc transferase (OGT) has proven to be a challenge,
especially because the diversity of published inhibitors is low. The large majority of available …
especially because the diversity of published inhibitors is low. The large majority of available …
New thiazolyl-isoxazole derivatives as potential anti-infective agents: design, synthesis, in vitro and in silico antimicrobial efficacy
MR Bhoye, A Shinde, ALN Shaikh… - Journal of …, 2024 - Taylor & Francis
Antimicrobial resistance threatens the efficacious prevention and treatment of infectious
diseases caused by microorganisms. To combat microbial infections, the need for new drug …
diseases caused by microorganisms. To combat microbial infections, the need for new drug …
Synthesis and characterization of thiazolidine-4-one compounds derived from chalcone and evaluation of the biological activity of some of them
ST Taha, MGA Karim, SS Jassim - Materials Today: Proceedings, 2022 - Elsevier
In this paper, chalcone [T1-T10] was synthesized from the reaction of (N-phenylacetamide or
N-(4-chlorophenyl) acetamide) with benzaldehyde and its aromatic substitutes using ethanol …
N-(4-chlorophenyl) acetamide) with benzaldehyde and its aromatic substitutes using ethanol …
[PDF][PDF] Synthesis and antimycobacterial screening of a novel series of α-amino acids containing thiazole linker
JL Nalawade, PC Mhaske, AD Shinde, AP Chavan… - Arkivoc, 2022 - arkat-usa.org
A small focused library of uncommon (S)-2-amino-3-(4-(((4-methyl-2-arylthiazol-5-yl) methyl)
amino) phenyl) propanoic acid (5a-e) and (S)-2-amino-3-(4-(((2-arylthiazol-4-yl) methyl) …
amino) phenyl) propanoic acid (5a-e) and (S)-2-amino-3-(4-(((2-arylthiazol-4-yl) methyl) …
Synthesis and antimicrobial activity of novel thiazolidinone derivatives
WO Alsulami, ZM Alamshany - platform.almanhal.com
The aim of this proposal is to synthesize and characterize a series of new novel
thiazolidinone derivatives and study their biological activities. These compounds are …
thiazolidinone derivatives and study their biological activities. These compounds are …