Development of a High-Throughput Screening Assay for Small-Molecule Inhibitors of Androgen Receptor Splice Variants

AE Monaghan, A Porter, I Hunter… - ASSAY and Drug …, 2022 - liebertpub.com
The role of the androgen receptor (AR) in the progression of prostate cancer (PCa) is well
established and competitive inhibition of AR ligand binding domain (LBD) has been the …