Facile and regioselective synthesis of new fluorinated [1, 2, 4]-triazolo [4, 3-a] pyrimidin-7 (1H)-one derivatives from fluorinated alkynes

B Jismy, H Allouchi, M Aweli, M Abarbri… - Journal of Fluorine …, 2020 - Elsevier
A mild, simple and efficient method for the regioselective synthesis of 3-substituted-1-phenyl
[1, 2, 4]-triazolo [4, 3-a] pyrimidin-7 (1H)-ones bearing a perfluoroalkyl group on position 5 is …

2-methylsulfanyl-6-polyfluoroalkyl-pyrimidin-4-ones: synthesis and nucleophilic substitution reactions

OG Khudina, YV Burgart, VI Saloutin - Chemistry of Heterocyclic …, 2014 - Springer
We have optimized the reaction conditions for the synthesis of 2-methylsulfanyl-6-polyfluoro-
alkylpyrimidin-4-ones. In particular the yield of trifluoromethyl-substituted heterocycle was …