Over the last two decades, transition-metal catalyzed C–H functionalization of indoles has
emerged as an area of extensive research and tremendous progress has been made in this …

A novel and versatile method for peri-C–H selenylation of aromatic compounds bearing
ketone groups, including chromones, xanthones, acridinones, quinolinones and …

Over the past decade, dioxazolones have been widely used as N-acylamide sources in
amidation processes of challenging substrates, typically employing precious transition …

With alanine as a transient directing group, Pd-catalyzed regioselective alkynylation at the
indole C4-position was successfully established in a good yield. The total synthesis of the …

A versatile and efficient method for the coupling of maleimides and indoles at the C7‐
position has been established under Rh (III) catalysis. The present protocol was compatible …

Aminoindoles are important synthetic intermediates to a broad range of bioactive molecules.
Transition metal‐catalyzed directed C− H amination is among the most straightforward route …

Regioselective direct functionalization of an indole benzenoid fragment has been a
significant challenge because of its inherently lower reactivity. In this report, we introduce a …

Multi-drug resistant Staphylococcus aureus infection is still a serious threat to global health.
Therefore, there is an urgent need to develop new antibacterial agents based on virulence …

The resistance of methicillin-resistant Staphylococcus aureus (MRSA) has augmented due
to the abuse of antibiotics, bringing about difficulties in the treatment of infection especially …

Heterocycle-braced cyclic peptides have demonstrated enhanced metabolic stability,
increased potency and selectivity. Here, we present a rapid synthesis method for …