Owing to the market competitiveness and urgent societal need, an optimum speed of drug
discovery is an important criterion for successful implementation. Despite the rapid ascent of …

The synthesis of substituted indoles has received great attention in the field of organic
synthesis methodology. C–H activation makes it possible to obtain a variety of designed …

The Rh (III)-catalyzed C–H oxidative alkylation of aniline derivatives with readily available
secondary allyl alcohols using a pyrimidine-directing group, leading to the production of β …

Rhodium (III)-catalyzed synthesis of indole derivatives has been realized via cascade
reaction of Csingle bondH alkylation/nucleophilic cyclization starting from readily available …

A ruthenium (II)-catalyzed redox-neutral synthesis of dihydroisoquinoline-fused
quinazolinone derivatives has been accomplished through the merger of C–H activation and …

The regioselective Rh (III)-catalyzed C–H amidation of aniline derivatives with dioxazolones
as an amidating reagent with a pyrimidine as a directing group leading to the production of …

Convenient, easily handled, laboratory friendly, robust approaches to afford synthetically
important organoboron compounds are currently of great interest to researchers. Among the …

An electrochemical approach to promote the ortho-C–H alkylation of (hetero) arenes via
rhodium catalysis under mild conditions is described. This approach features mild conditions …

A versatile rhodium-catalyzed/copper-mediated C–H/C–C activation and cascade
annulation reaction was described to form 2-arylindole derivatives. Highly selective C–C …

Non‐activated allyl alcohols are utilized as allylating agent for thiocarbamate‐directed
allylation of pyrrole and indole. The synthetic methodology is accompanied by advantages …