Unsaturated polyfluoroalkyl ketones in the synthesis of nitrogen-bearing heterocycles

AY Rulev, AR Romanov - RSC advances, 2016 - pubs.rsc.org
Unsaturated polyfluoroalkyl ketones in the synthesis of nitrogen-bearing heterocycles - RSC
Advances (RSC Publishing) DOI:10.1039/C5RA23759A Royal Society of Chemistry View …

[PDF][PDF] Preparation of α, β-unsaturated trifluoromethylketones and their application in the synthesis of heterocycles

VG Nenajdenko, ES Balenkova - Arkivoc, 2011 - arkat-usa.org
Preparation of α,β-unsaturated trifluoromethylketones and their application in the synthesis of
heterocycles Page 1 Reviews and Accounts ARKIVOC 2011 (i) 246-328 Page 246 ©ARKAT-USA …

Structure-Based Virtual Screening and In Vitro Evaluation of New Trypanosoma cruzi Cruzain Inhibitors

V Herrera-Mayorga, EE Lara-Ramírez… - International journal of …, 2019 - mdpi.com
Chagas disease (CD), or American trypanosomiasis, causes more than 10,000 deaths per
year in the Americas. Current medical therapy for CD has low efficacy in the chronic phase …

Heterocyclization of N-(1-chloro-2, 2, 2-trifluoroethylidene) carbamates with β-enaminoesters—a novel synthetic strategy to functionalized trifluoromethylated …

VA Sukach, VM Tkachuk, EB Rusanov… - Tetrahedron, 2012 - Elsevier
Heterocyclization of N-(1-chloro-2,2,2-trifluoroethylidene)carbamates with β-enaminoesters—a
novel synthetic strategy to functionalized trifluoromethylated pyrimidines - ScienceDirect …

Chemo-and regioselective reactions of 5-bromo enones/enaminones with pyrazoles

PA Moraes, MM Lobo, MA Marangoni… - Organic & …, 2019 - pubs.rsc.org
Reaction of 5-bromo enones with pyrazoles provided a series of unexpected N, O-aminal
derivatives, through a 1, 4-conjugated addition at the β-carbon of the 5-bromo enones …

Synthesis and structural study of N-methyl-2-methylthiopyrimidine derivatives from trihalomethylated enones.

N Zanatta, CC Madruga, PC Marisco… - Journal of …, 2010 - search.ebscohost.com
Abstract < GRAPHIC> </GRAPHIC> The synthesis and chemoselective study of a
novel series N-methyl-2-methylthio-tetrahydropyrimidines and or N-methyl-2 …

An Environmentally Benign Multicomponent Synthesis of Some Novel 2‐Methylthio Pyrimidine Derivatives Using MCM‐41‐NH2 as Nanoreactor and Nanocatalyst

S Rostamizadeh, M Nojavan - Journal of Heterocyclic …, 2014 - Wiley Online Library
Some novel 4‐amino‐6‐aryl‐2‐methylthio pyrimidine‐5‐carbonitrile derivatives were
synthesized through a one‐pot three‐component reaction of an aldehyde, malononitrile, and …

Regioselective Reactions of Ethyl (4, 5-Dihydrofuran-3-yl)-2-oxoacetate and Ethyl 2-(3, 4-Dihydro-2H-pyran-6-yl)-2-oxoacetate with 1-Unsubstituted Aminoazoles

OO Stepaniuk, VO Matvienko, IS Kondratov… - …, 2012 - thieme-connect.com
Abstract The reactions of ethyl (4, 5-dihydrofuran-3-yl)-2-oxoacetate and ethyl 2-(3, 4-
dihydro-2H-pyran-6-yl)-2-oxoacetate, as 1, 3-bielectrophiles, with N-unsubstituted 5 …

Highly Chemoselective Synthesis of 6‐Alkoxy‐1‐alkyl (aryl)‐3‐trifluoroacetyl‐1, 4, 5, 6‐tetrahydropyridines and 1‐Alkyl (aryl)‐6‐amino‐3‐trifluoroacetyl‐1, 4, 5, 6 …

N Zanatta, L da S. Fernandes, FM Nachtigall… - 2009 - Wiley Online Library
A simple and highly chemoselective method for the synthesis of a large series of novel 6‐
alkoxy‐1‐alkyl (aryl)‐3‐trifluoroacetyl‐1, 4, 5, 6‐tetrahydropyridines and 1‐alkyl (aryl)‐6 …

Synthetic routes to 1, 4, 5, 6-tetrahydropyrimidines: An overview and recent advances

A Bhattacharyya - Current Organic Chemistry, 2019 - ingentaconnect.com
Partially reduced heterocyclic compounds such as 1, 4, 5, 6-tetrahydropyrimidines are often
found to possess interesting pharmacological properties. Yet, the synthetic routes towards …