Synthesis and biological evaluation of resveratrol amide derivatives as selective COX-2 inhibitors

M Xin, H Wu, Y Du, S Liu, F Zhao, X Mou - Chemico-Biological Interactions, 2023 - Elsevier
Selective COX-2 inhibitors have been considered to be reliable alternatives to tNSAIDs, but
most of them were withdrawn from the market due to their risk of heart attack and stroke …

[PDF][PDF] QSAR study of benzylidene hydrazine benzamides derivatives with in vitro anticancer activity against human lung cancer cell line A459

GS Putra, MI Sulistyowaty, TA Yuniarta… - Journal of Pharmacy & …, 2023 - academia.edu
Context: In the last decade, resistance to epidermal growth factor receptor-tyrosine kinase
inhibitors (EGFR-TKIs) in lung cancer cases has been widespread. The discovery and …

Hansch analysis by QSAR model of curcumin and eight of its transformed derivatives with antimicrobial activity against Staphylococcus aureus

D Kesuma, GS Putra, Y Yahmin… - … of Pharmacy & …, 2024 - repository.ubaya.ac.id
Context: In the last decade, antimicrobial resistance cases have been widespread. The
discovery and development of new drugs need to be done to overcome the case. Some …

Atom-economical synthesis, antimicrobial assessment, and molecular dynamics of indole-derived peptidomimetics for improved therapeutic insights

S Sebastian, Y Rohila, S Prakash, A Kumar… - Journal of Molecular …, 2024 - Elsevier
The emergence of multi-drug resistant strains spanning bacteria, fungi, viruses, and
parasites poses a severe threat to public health and the economy. Tackling antimicrobial …

[HTML][HTML] Curcumin derivatives against Staphylococcus aureus

D Kesuma, GS Putra, Y Yahmin, S Sumari, AO Putri… - jppres.com
Context: In the last decade, antimicrobial resistance cases have been widespread. The
discovery and development of new drugs need to be done to overcome the case. Some …

[HTML][HTML] Benzylidene hydrazine benzamide derivatives QSAR study

Context: In the last decade, resistance to epidermal growth factor receptor-tyrosine kinase
inhibitors (EGFR-TKIs) in lung cancer cases has been widespread. The discovery and …