In silico molecular docking against C-KIT tyrosine kinase and ADME studies of 3-ethyl-2-(2, 3, 4-trifluoro-phenylimino)-thiazolidin-4-one derivatives

SD Kadam, D Mammen, DS Kadam, SG Patil - 2023 - indianjournals.com
Thiazolidin-4-one derivatives have been hailed as “wonder nucleus” due to their profound
biological activities. A number of derivatives with variable functional groups attached to the …

Synthesis, antimicrobial properties and in silico studies of aryloxyacetic acid derivatives with hydrazone or thiazolidine-4-one scaffold

S Şenkardeş, D Kart, B Bebek, MG Gündüz… - Journal of …, 2023 - Taylor & Francis
In this work, twenty hydrazide-hydrazone and 4-thiazolidinone derivatives were synthesized
starting from m-cresol. Antimicrobial evaluation was carried out by microdilution method …

[PDF][PDF] In silico molecular docking against-KIT tyrosine kinase and ADME studies of 4-thiazolidinone derivatives

D Kadam, S Patil, D Mammen, S Kadam, V More - Journal of Applied …, 2023 - sid.ir
Archive of SID.ir Archive of SID.ir Page 1 2023, Volume 3, Issue 1 13 2021, Volume 2, Number
1 Original Article In Silico Molecular Docking Againstc-KIT Tyrosine Kinase and ADME Studies …

Novel fluorinated thiazolidin-4-one derivatives: synthesis and anti-cancer potential against HepG2 and HCT116 cell lines

SD Kadam, D Mammen, V Zunjar… - Australian Journal of …, 2024 - CSIRO Publishing
A novel synthetic route has been designed to introduce fluorine functionality into a series of
compounds containing thiazolidin-4-one rings. These compounds were synthesised from …

Evaluation of 3-Ethyl-5-fluoro-2-phenylimino-thiazolidin-4-one derivatives: Molecular docking against kinase protein and ADME studies

SD Kadam, D Mammen, LB Nikam… - Research Journal of …, 2024 - search.proquest.com
A number of new compounds have been synthesized by the authors containing fluorinated
thiazolidin-4-one ring. With the aim to assess the anti-cancer potential of all the synthesized …

Synthesis, characterization and evaluation of in vitro anticancer potential of novel fluorinated 5-benzylidene-3-ethyl-2-(2-methyl-3-trifluoromethyl-phenylimino) …

SD Kadam, D Mammen, LB Nikam, RR Bagul - 2024 - nopr.niscpr.res.in
A set of novel 5-benzylidene-3-ethyl-2-(2-methyl-3-trifluoromethyl-phenylimino)-thiazolidin-4-
one derivatives have been synthesized by Knoevenagel reaction via both conventional as …

Synthesis and biological evaluation of new 4-thiazolidinone derivatives of flurbiprofen

P Suzgun, S Şenkardeş, M Gurboga… - Organic …, 2023 - avesis.marmara.edu.tr
In this study, the synthesis and characterization of 2-(2-fluorobiphenyl-4-yl)-N'-[(substituted
methylene] propanehydrazides (3a-s) and 2-(2-fluoro-[1, 1'-biphenyl]-4-yl)-N-(5-methyl-2 …

Synthesis of sulfonamides bearing 1, 3, 5-triarylpyrazoline and 4-thiazolidinone moieties as novel antimicrobial agents

TD Thach, TTV Le, HTA Nguyen, CH Dang… - Journal of the Serbian …, 2020 - shd-pub.org.rs
Two series of sulfonamides were synthesized from 4-hydrazinylbenzenesulfonamide as the
key starting material. 1, 3, 5-Triarylpyrazoline sulfonamides (2a–i) were obtained by …