Recent advances in the synthesis of pyrrolo [1, 2-a] indoles and their derivatives

YG Shelke, PE Hande, SJ Gharpure - Organic & Biomolecular …, 2021 - pubs.rsc.org
The pyrrolo [1, 2-a] indole unit is a privileged heterocycle found in numerous natural
products and has been shown to exhibit diverse pharmacological properties. Thus, recent …

Isoindolinone Synthesis via One‐Pot Type Transition Metal Catalyzed C− C Bond Forming Reactions

R Savela, C Méndez‐Gálvez - Chemistry–A European Journal, 2021 - Wiley Online Library
Isoindolinone structure is an important privileged scaffold found in a large variety of naturally
occurring as well as synthetic, biologically and pharmaceutically active compounds. Owing …

Sustainable preparation of photoactive indole-fused tetracyclic molecules: a new class of organophotocatalysts

J Bae, N Iqbal, HS Hwang, EJ Cho - Green Chemistry, 2022 - pubs.rsc.org
Efficient and sustainable preparation of photoactive indole-fused tetracyclic molecules and
their application as organophotocatalysts have been developed. Additive-free and air stable …

Palladium-catalyzed cross-dehydrogenative coupling of (hetero) arenes

G Albano - Organic Chemistry Frontiers, 2024 - pubs.rsc.org
Organic compounds based on (hetero) aryl scaffolds are systems with a wide range of
application, from pharmaceuticals and agrochemicals to semiconducting materials for …

Rhodium-Catalyzed NH-Indole-Directed C–H Carbonylation with Carbon Monoxide: Synthesis of 6H-Isoindolo[2,1-a]indol-6-ones

Q Huang, Q Han, S Fu, Z Yao, L Su… - The Journal of …, 2016 - ACS Publications
An efficient synthesis of 6 H-isoindolo [2, 1-a] indol-6-ones through rhodium-catalyzed NH-
indole-directed C–H carbonylation of 2-arylindoles with carbon monoxide has been …

Steering Site‐Selectivity in Transition Metal‐Catalyzed C− H Bond Functionalization: the Challenge of Benzanilides

R Gramage‐Doria - Chemistry–A European Journal, 2020 - Wiley Online Library
Selective C− H bond functionalization catalyzed by metal complexes have completely
revolutionized the way in which chemical synthesis is conceived nowadays. Typically, the …

One-Step Synthesis of Isoindolo[2,1-a]indol-6-ones via Tandem Pd-Catalyzed Aminocarbonylation and C–H Activation

T Čarný, M Markovič, T Gracza… - The Journal of Organic …, 2019 - ACS Publications
A unified catalytic system for tandem Pd-catalyzed carbonylation and C–C cross-coupling
via C–H activation was designed. The proposed cascade reaction allows a facile one-step …

The synthesis of N‐benzoylindoles as inhibitors of rat erythrocyte glucose‐6‐phosphate dehydrogenase and 6‐phosphogluconate dehydrogenase

S Bayindir, Y Temel, A Ayna… - Journal of biochemical …, 2018 - Wiley Online Library
Abstract Glucose‐6‐phosphate dehydrogenase (G6PD) and 6‐phosphogluconate
dehydrogenase (6PGD) play an important function in various biochemical processes as they …

Intramolecular Carbonylative C–H Functionalization of 1,2,3‐ Triazoles for the Synthesis of Triazolo[1,5‐a]indolones

C Veryser, G Steurs, L Van Meervelt… - Advanced Synthesis …, 2017 - Wiley Online Library
This study presents a synthesis of 4H‐[1, 2, 3] triazolo [1, 5‐a] indol‐4‐ones. The key step in
the synthesis of this new heterocyclic scaffold is an intramolecular cyclization via an …

[HTML][HTML] Palladium-catalyzed intramolecular tandem dearomatization of indoles for the synthesis of tetracyclic indolines

SB Duan, XJ Gao, HY Zhang, CC Lu, J Zhao… - Arabian Journal of …, 2021 - Elsevier
A highly diastereoselective, atom-economical, and palladium-catalyzed Heck protocol for
the assembly of structurally diverse indoline scaffolds with vicinal tertiary as well as …