Click chemistry: 1, 2, 3‐triazoles as pharmacophores

SG Agalave, SR Maujan… - Chemistry–An Asian …, 2011 - Wiley Online Library
Abstract The copper (I)‐catalyzed 1, 2, 3‐triazole‐forming reaction between azides and
terminal alkynes has become the gold standard of 'click chemistry'due to its reliability …

Synthesis of quinoline coupled [1, 2, 3]-triazoles as a promising class of anti-tuberculosis agents

KK Kumar, SP Seenivasan, V Kumar, TM Das - Carbohydrate research, 2011 - Elsevier
A series of quinoline coupled 1, 2, 3-triazoles compounds have been synthesized by 'click
chemistry'from azidomethyl quinoline with different alkynes. The efficiency and fidelity of the …

Mechanostereoselective one-pot synthesis of functionalized head-to-head cyclodextrin [3] rotaxanes and their application as magnetic resonance imaging contrast …

JW Fredy, J Scelle, G Ramniceanu, BT Doan… - Organic …, 2017 - ACS Publications
A versatile, five-component, one-pot synthesis of cyclodextrin (CD)[3] rotaxanes using
copper-catalyzed azide–alkyne cycloaddition has been developed. Head-to-head [3] …

Design and synthesis of sugar-triazole low molecular weight gels as mercury ion sensor

A Hemamalini, TM Das - New Journal of Chemistry, 2013 - pubs.rsc.org
A series of gel forming symmetrical bis-sugar-triazoles has been developed for the
recognition of Hg2+ ions. Preferential interaction of Hg2+ ions with organogelator based …

Chemical Synthesis of N-Aryl Glycosides

MY Fosso, VPN Nziko, CWT Chang - Journal of Carbohydrate …, 2012 - Taylor & Francis
Along with the O-and C-aryl glycosides, N-aryl glycosides represent an important class of
carbohydrate and heterocyclic aryl conjugates that possess diverse applications and …

FACE-selective fluorogenic cycloaddition reaction between coumarin azides and sugar terminal alkynes: an experimental and computational study

R Rajaganesh, P Ravinder, V Subramanian… - Carbohydrate …, 2011 - Elsevier
Copper catalyzed azide–alkyne cycloaddition reaction (CuAAC) of non-fluorescent
coumarin azides and sugar terminal alkynes afforded intense fluorescent 1, 2, 3-triazoles in …

Synthesis of N1 and N2 coumarin substituted 1,2,3-triazole isomers via click chemistry approach

D Shamala, K Shivashankar, Chandra… - Synthetic …, 2016 - Taylor & Francis
The synthesis of N1 and N2 coumarin substituted 1, 2, 3-triazole isomers from terminal
alkynes, sodium azide, and 4-bromomethylcoumarins in the presence of triethylamine as a …

Rational Design of Heterocyclic Moieties Incorporated in [1, 2, 3] Sugar‐Triazole Derivatives for Antioxidant Studies

VR Jenifer, P Muthuvel, TM Das - ChemistrySelect, 2021 - Wiley Online Library
Reaction of heterocyclic azides with sugar alkyne under copper catalyzed 1, 3‐dipolar
cycloaddition reaction resulted in the formation of triazoles in 64–90% of yield. Existence of …

Research on the structure–surface adsorptive activity relationships of triazolyl glycolipid derivatives for mild steel in HCl

HL Zhang, XP He, Q Deng, YT Long, GR Chen… - Carbohydrate …, 2012 - Elsevier
Triazolyl glycolipid derivatives constructed via CuI-catalyzed azide-alkyne 1, 3-dipolar
cycloaddition reaction (Cue-AAC) represent a new range of carbohydrate-based scaffolds …

Studies on the synthesis and the antimicrobial and antioxidant activities of a novel class of fluorescein-based glycosides

M Rajasekar, R Jegadeesh, N Raaman, TM Das - Carbohydrate research, 2011 - Elsevier
Facile glycosylation of a fluorescein diol derivative with per-O-acetyl/benzoyl sugar
derivatives using BF3· Et2O catalyst resulted in the formation of the expected glycosides in …