Recently, owing to their special spatial structures, peptide-based macrocycles have shown
tremendous promise and aroused great interest in multidisciplinary research ranging from …

Enzyme‐triggered macrocyclization and in situ self‐assembly of small molecules into
nanoparticles has shown promise to design activatable probes for molecular imaging …

Bicyclic peptides possess superior properties for drug discovery; however, their chemical
synthesis is not straightforward and often neither biocompatible nor fully orthogonal to all …

Multifunctional porphyrin–peptide conjugates with different propensities for self‐assembly
into various supramolecular nanoarchitectures play important roles in advanced materials …

Tumor-targeted near-infrared (NIR) fluorescence imaging by using NIR fluorescent probes
has attracted extensive attentions in the field of tumor imaging and is becoming an attractive …

Polyfluorinated aromatic reagents readily react with thiolates via nucleophilic aromatic
substitution (SNAr) and provide excellent scaffolds for peptide cyclisation. Here we report a …

Corroles have attracted increasing research interests in recent decades owing to their
unique properties over porphyrins. However, the relatively inefficient and tedious synthetic …

Hybrid sequences comprising a peptide with several Cys residues and an aromatic foldamer
helix with several chloroacetamide functions at its surface were synthesized. Such products …

Cyclen‐peptide bioconjugates are usually prepared in multiple steps that require individual
preparation and purification of the cyclic peptide and hydrophilic cyclen derivatives. An …

Combination of cysteine-containing peptides with electrophiles provides efficient access to
cyclo-organopeptides. However, there are no routes to intrinsically fluorescent cyclo …