Synthesis and biological evaluation of novel acyclic and cyclic glyoxamide based derivatives as bacterial quorum sensing and biofilm inhibitors

S Nizalapur, O Kimyon, E Yee… - Organic & …, 2017 - pubs.rsc.org
Bacteria regulate the expression of various virulence factors and processes such as biofilm
formation through a chemically-mediated communication mechanism called quorum …

Magnetic metal–organic framework CoFe2O4@ SiO2@ IRMOF-3 as an efficient catalyst for one-pot synthesis of functionalized dihydro-2-oxopyrroles

JN Zhang, XH Yang, WJ Guo, B Wang, ZH Zhang - Synlett, 2017 - thieme-connect.com
A magnetic metal–organic framework-based catalyst CoFe 2 O 4@ SiO 2@ IRMOF-3 was
prepared and identified as an efficient catalyst for the synthesis of a variety of functionalized …

Synthesis, in Silico Study and Biological Evaluation of N‐(Benzothiazol/Thiazol‐2‐yl) benzamide Derivatives as Quorum Sensing Inhibitors against Pseudomonas …

N Sharma, N Srivastava, A Kaushal… - Chemistry & …, 2023 - Wiley Online Library
The development of bacterial resistance to chemical therapy poses a severe danger to
efficacy of treating bacterial infections. One of the key factors for resistance to antimicrobial …

Preparation of 3, 5-diarylsubstituted 5-hydroxy-1, 5-dihydro-2 H-pyrrol-2-ones via base-assisted cyclization of 3-cyanoketones

NA Aksenov, DA Aksenov, IA Kurenkov, AV Aksenov… - RSC …, 2021 - pubs.rsc.org
A convenient preparative method is developed allowing for expeditious assembly of 3, 5-
diarylsubstituted 5-hydroxy-1, 5-dihydro-2H-pyrrol-2-ones from routinely available …

Strategies to access γ-hydroxy-γ-butyrolactams

MID Mardjan, JL Parrain, L Commeiras - Synthesis, 2018 - thieme-connect.com
α, β-Unsaturated γ-hydroxy-γ-butyrolactams are of a great interest due to their presence in
designed pharmaceutical molecules and numerous natural products displaying a broad …

Synthesis, Biological Evaluation and in Silico Study of N‐(2‐and 3‐Pyridinyl) benzamide Derivatives as Quorum Sensing Inhibitors against Pseudomonas aeruginosa

N Sharma, N Srivastava, B Devi, L Kumar… - Chemistry & …, 2023 - Wiley Online Library
The effectiveness of treating bacterial infections is seriously threatened by the emergence of
bacterial resistance to chemical treatment. Growth of microbes in biofilm is one of the main …

Total synthesis, structural revision and biological evaluation of γ-elemene-type sesquiterpenes

C Yuan, S Zhong, X Li, Y Wang, MM Xun… - Organic & Biomolecular …, 2018 - pubs.rsc.org
Total synthesis and absolute configuration confirmation of γ-elemene-type sesquiterpenes,
which possess vast potential for biological activities, was investigated based on a …

Synthesis of new dihydropyrrol-2-one derivatives bearing sulfonamide groups and studies their antibacterial activity

M Bavadi, K Niknam, M Gharibi - Monatshefte für Chemie-Chemical …, 2017 - Springer
A novel series of dihydropyrrol-2-one compounds bearing sulfonamide groups were
synthesized and assayed for in vitro antibacterial activity against Staphylococcus aureus …

Quorum Sensing Inhibition: Current Advances of the Natural Antimicrobial Agents

M Asif, M Imran - Russian Journal of Bioorganic Chemistry, 2019 - Springer
The misuses of antimicrobials in infectious diseases have led to the progress of extensive
resistance in the infectious organisms. The failure of accessible antimicrobials to control …

[PDF][PDF] Design, synthesis and biological evaluation of novel glyoxamide based antibacterial agents

S Nizalapur - 2018 - scholar.archive.org
dspace cover page Page 1 Design, synthesis and biological evaluation of novel glyoxamide
based antibacterial agents Author: Nizalapur, Shashidhar Publication Date: 2018 DOI: https://doi.org/10.26190/unsworks/20258 …