Heterocyclic alkenes represent an important class of reactive feedstock and valuable
synthons for the synthesis of biologically important heterocyclic scaffolds. Although …

Selective editing of the benzenoid C− H bonds (C4− C7) in indoles/indolines has received
great interest because functionalized indoles/indolines are featured in many marketed drugs …

The indole scaffold is a ubiquitous and useful substructure, and extensive investigations
have been conducted to construct the indole framework and/or realize indole modification …

We report the synthesis of carbazole-based unnatural α-amino acid and non-α-amino acid
derivatives via a Pd (II)-catalyzed bidentate directing group 8-aminoquinoline-aided β-C …

Rhodium-catalyzed diverse tandem twofold C–H bond activation reactions of para-olefin-
tethered arenes have been realized, with unsaturated reagents such as internal alkynes …

Transition‐metal‐catalyzed C− H functionalization is one of the fascinating scientific fronts in
organic synthesis for the formation of conjugated arenes and has emerged as a benchmark …

Here we report a protocol to synthesize diversiform fluorinated isocryptolepine analogues
with potential biological activities in one step via directed C-2 and C-3 dual C–H …

Cu-catalyzed cross-dehydrogenative coupling of the C7 C–H bond of indolines with
sulfoximines has been accomplished. The reaction can be extended to the cross …

C8-Substituted quinoline (QN) and 1, 2, 3, 4-tetrahydroquinoline (THQ) scaffolds are
featured in numerous bioactive compounds and natural products. Appreciable efforts have …

A nickel-catalyzed site-selective tandem cyclization of 1, 6-diynes with substituted indolines
or indoles through consecutive dual C–H bond activation is described. In the reaction …