[HTML][HTML] Nicotine-sensitive acetylcholine receptors are relevant pharmacological targets for the control of multidrug resistant parasitic nematodes

CL Charvet, F Guégnard, E Courtot, J Cortet… - International Journal for …, 2018 - Elsevier
The control of parasitic nematodes impacting animal health relies on the use of broad
spectrum anthelmintics. However, intensive use of these drugs has led to the selection of …

Asymmetric cross-coupling of alkyl, alkenyl and (hetero) aryl nucleophiles with racemic allyl halides

P Schäfer, M Sidera, T Palacin… - Chemical …, 2017 - pubs.rsc.org
Single enantiomer molecules are important for the pharmaceutical and agrochemical
industries and increasingly so in materials science. Most strategies to obtain …

Potential modulating effect of the Ascaris suum nicotinic acetylcholine receptor (nAChR) by compounds GSK575594A, diazepam and flumazenil discovered by …

S Stevanovic, DS Marjanović, SM Trailović… - Molecular and …, 2021 - Elsevier
Parasitic infections are a widespread health problem and research of novel anthelmintic
compounds is of the utmost importance. In this study we performed a virtual screening …

Mechanism of action of drugs with activity against multicellular parasites

C Giordani, GH Marin, D Perez, AL Soraci, J Errecalde - 2017 - ri.conicet.gov.ar
Parasiticides have been the most valuable weapons to combat parasites for almost half a
century, constituting more than 50% of veterinary pharmaceuticals and a good part of the …

[HTML][HTML] Desarrollo de fármacos antihelmínticos: actualización de candidatos a fármacos y dianas terapéuticas en el manejo de las geohelmintiasis

AM Uribe Herrera, AP Rojas, P Reyes Harker… - Revista Med, 2022 - scielo.org.co
se estima que 1500 millones de personas en el mundo están infectadas por algún
geohelminto. La disminución de la eficacia de los medicamentos antihelmínticos utilizados …

[PDF][PDF] IJP: Drugs and Drug Resistance

CL Charvet, F Guégnard, E Courtot, J Cortet, C Neveu - researchgate.net
The control of parasitic nematodes impacting animal health relies on the use of broad
spectrum anthelmintics. However, intensive use of these drugs has led to the selection of …

МЕХАНИЗМ ДЕЙСТВИЯ ЛЕКАРСТВ, ОБЛАДАЮЩИХ АКТИВНОСТЬЮ ПРОТИВ МНОГОКЛЕТОЧНЫХ ПАРАЗИТОВ

C Giordani, GH Marin, D Pérez, A Soraci, J Errecalde - Паразитология, 2017 - elibrary.ru
Средства, убивающие паразитов (паразитициды), служили наиболее доступным
оружием в борьбе с паразитами почти в течение полувека, составляя более половины …

Enantioselective synthesis of chiral building blocks with non-stabilized nucleophiles

P Schäfer - 2017 - ora.ox.ac.uk
This thesis describes the combination of non-stabilized nucleophiles and prochiral/racemic
electrophiles in transition metal catalyzed asymmetric transformations. These …

[引用][C] Síntesis de compuestos neo-nicotínicos con afinidad a los receptores nicotínicos α4β2 ya los transportadores de serotonina y dopamina

JP González-Gutiérrez - 2020