Guanidinium-functionalized flexible azaproline transporter for efficient intracellular delivery of proapoptotic peptide and PDL1 antisense morpholino oligo in human …
Cell-penetrating peptides (CPPs) are structurally diverse sophisticated tools endowed with
high arginine content, amphipathicity, and well-adopted suitable secondary structures …
high arginine content, amphipathicity, and well-adopted suitable secondary structures …
Stereoselective synthesis of (R)-and (S)-1, 2-diazetidine-3-carboxylic acid derivatives for peptidomimetics
M Nutter, H Stone, M Shipman… - Organic & Biomolecular …, 2024 - pubs.rsc.org
The stereoselective synthesis of both enantiomers of N-protected 1, 2-diazetidine-3-
carboxylic acid (aAze) from homochiral glycidol is described. Orthogonal protection of this …
carboxylic acid (aAze) from homochiral glycidol is described. Orthogonal protection of this …
Synthesis of Fmoc-protected amino alcohols via the Sharpless asymmetric aminohydroxylation reaction using FmocNHCl as the nitrogen source
R Moreira, M Diamandas, SD Taylor - The Journal of Organic …, 2019 - ACS Publications
The aminohydroxylation of various alkenes using FmocNHCl as a nitrogen source is
reported. In general, in the absence of a ligand, the reaction provided racemic Fmoc …
reported. In general, in the absence of a ligand, the reaction provided racemic Fmoc …
Synthesis of a tripeptide biomarker of exposure to sulfur mustard for support of OPCW biomedical proficiency tests
VV Abzianidze, YV Chelusnova, GV Karakashev… - Mendeleev …, 2021 - Elsevier
Synthesis of a tripeptide biomarker of exposure to sulfur mustard for support of OPCW
biomedical proficiency tests - ScienceDirect Skip to main contentSkip to article Elsevier logo …
biomedical proficiency tests - ScienceDirect Skip to main contentSkip to article Elsevier logo …
Synthesis and Study of the Cyclic Lipopeptide Antibiotics Daptomycin and A54145
R Moreira - 2022 - uwspace.uwaterloo.ca
Daptomycin (dap) is a clinical antibiotic used to treat infections with multi-drug resistant
Gram-positive bacteria. Despite nearly 20 years of clinical use, the action mechanism of this …
Gram-positive bacteria. Despite nearly 20 years of clinical use, the action mechanism of this …
δ-Azaproline: A versatile tool to design pseudopeptides by its incorporation via Nε or Nδ atoms
O Ovdiichuk, L Flauder, E Humbert-Voss… - Tetrahedron …, 2019 - Elsevier
Abstract δ-Azaproline, a bis-nitrogen proline, has been incorporated in pseudotripeptides of
the type Xaa 1-δazaPro-Xaa 3. Peptide elongation via both nitrogen atoms has been …
the type Xaa 1-δazaPro-Xaa 3. Peptide elongation via both nitrogen atoms has been …
[引用][C] Desarrollo y diversificación de sistemas catalíticos basados en hidrozonas. Aplicaciones en catálisis asimétrica
S Alberca Manzano - 2023