Hydroxyphosphonates have attracted considerable attention as biologically active
compounds, enzyme inhibitors, and drugs. Over the last few years significant interest in the …

Published data on the synthesis, absolute configurations and biological properties of chiral
hydroxy phosphonates are generalised and described systematically. Examples of …

This review presents a comprehensive account of methods which are commonly applied for
the synthesis of α-aminophosphonic acids. In the following order, protocols based on the …

The 1, 3-oxazolidin-2-one nucleus is a popular heterocycle framework in synthetic organic
chemistry, as well as in medicinal chemistry. This paper deals with the huge number of …

Abstract α‐Amino phosphonic acid derivatives are considered to be the most important
structural analogues of α‐amino acids and have a very wide range of applications. However …

Due to their use as analogues of aminoacids, aminophosphonates have attracted
considerable attention in the recent years. These compounds show a wide range of …

α-Isothiocyanato phosphonates are first used as nucleophiles to react with aldehydes for the
asymmetric synthesis of β-hydroxy-α-amino phosphonic acid derivatives. The process is …

A versatile approach for the synthesis of both protected enantiomers of aziridine 2-
phosphonates for use as chiral synthons has been developed. The aziridines arise from …

Syntheses of 5-phosphono-2-oxazolidinones and 5-phosphono-2-imidazolidinones were
achieved from the corresponding 1-vinyl-2-phosphonoaziridines. Regioselective aziridine …

An efficient, diastereoselective synthesis of 5-substituted (2-thioxo-imidazolidin-4-yl)
phosphonic acid diethyl esters from metallated diethyl isothiocyanatomethylphosphonate …