Synthesis and biological activity of 4-thiazolidinones, thiosemicarbazides derived from diflunisal hydrazide

G Küçükgüzel, A Kocatepe, E De Clercq… - European journal of …, 2006 - Elsevier
Two novel series of 4-thiazolidinone derivatives, namely 2′, 4′-difluoro-4-
hydroxybiphenyl-3-carboxylic acid [2-(5-nitro-2-furyl/substituted phenyl)-4-thiazolidinone-3 …

Sulfonamide-1, 2, 4-triazole derivatives as antifungal and antibacterial agents: Synthesis, biological evaluation, lipophilicity, and conformational studies

IR Ezabadi, C Camoutsis, P Zoumpoulakis… - Bioorganic & Medicinal …, 2008 - Elsevier
A series of 10 new 5-[2-(substituted sulfamoyl)-4, 5-dimethoxy-benzyl]-4aryl-s-triazole-3-
thiones were synthesized and evaluated for in vitro antifungal and antibacterial activity. All …

Synthesis and antimicrobial activity of 4-phenyl/cyclohexyl-5-(1-phenoxyethyl)-3-[N-(2-thiazolyl) acetamido] thio-4H-1, 2, 4-triazole derivatives

G Turan-Zitouni, ZA Kaplancıklı, MT Yıldız… - European journal of …, 2005 - Elsevier
The increasing clinical importance of drug-resistant fungal and bacterial pathogens has lent
additional urgency to microbiological research and new antimicrobial compound …

Clubbed triazoles: a novel approach to antitubercular drugs

M Shiradkar, GVS Kumar, V Dasari, S Tatikonda… - European journal of …, 2007 - Elsevier
In last few decades, though significant progress has been made in the treatment and control
strategies of tubercular infections by introducing new diagnostic and monitoring tools and …

Synthesis and antimicrobial activity of some 1, 2, 4-triazole-3-mercaptoacetic acid derivatives

N Ulusoy, A Gürsoy, G Ötük - Il Farmaco, 2001 - Elsevier
Ethyl 5-(2-furyl)-4-ethyl-1, 2, 4-triazole-3-mercaptoacetate (2), 5-(2-furyl)-4-ethyl-1, 2, 4-
triazole-3-mercaptoacetic acid hydrazide (3) and a series of new N-alkylidene/arylidene-5-(2 …

Synthesis and biological evaluation of potent antifungal agents

A Geronikaki, M Fesatidou, V Kartsev… - Current topics in …, 2013 - ingentaconnect.com
The last two decades are characterized by major increases in the incidence of systemic
fungal infections caused by the yeast Candida albicans, particularly in immunocompromised …

Synthesis and antimycobacterial activity of [5-(pyridin-2-yl)-1, 3, 4-thiadiazol-2-ylthio] acetic acid arylidene-hydrazide derivatives

MG Mamolo, V Falagiani, D Zampieri, L Vio, E Banfi - Il Farmaco, 2001 - Elsevier
[5-(Pyridin-2-yl)-1, 3, 4-thiadiazol-2-ylthio] acetic acid arylidene-hydrazide derivatives were
synthesized and tested for their in vitro antimycobacterial activity. Some compounds showed …

Synthesis and biological evaluation of indole containing derivatives of thiosemicarbazide and their cyclic 1, 2, 4-triazole and 1, 3, 4-thiadiazole analogs

A Varvaresou, A Tsantili-Kakoulidou… - …, 2000 - thieme-connect.com
New indolic derivatives of thiosemicarbazides and some cyclic l, 2, 4-triazol-5-thione
analogs were synthesized. The newly synthesized compounds as well as some indole …

Insight into the synthesis, biological impact and convenient routes of hydrazonoyl halides for synthesis of novel bioactive heterocycles: Mini-review

SA Osman, MA Abdallah, H Bassiony… - Egyptian Journal of …, 2023 - journals.ekb.eg
The present survey review focuses on the synthetic methods of hydrazonoyl halides
published during the past 20 years. The review covers also the pharmaceutical and …

Efficient synthesis of novel 1, 2, 4-triazole fused acyclic and 21–28 membered macrocyclic and/or lariat macrocyclic oxaazathia crown compounds with potential …

NSAM Khalil - European journal of medicinal chemistry, 2010 - Elsevier
Versatile simple efficient routes with good to excellent yields towards different functionalized
1, ω-bis (1, 2, 4-triazoles), 21–28 membered 1, 2, 4-triazole fused macrocyclic and/or lariat …