Rhodanines are accepted as advantaged heterocycles in medicinal chemistry as one of the
4-thiazolidinones subtypes. The aim of this paper is to analyze the features of rhodanine and …

The genus Mycobacterium comprises not only the deadliest of bacterial pathogens,
Mycobacterium tuberculosis, but several other pathogenic species, including M. avium and …

Staphylococcus aureus is a Gram-positive bacterium that has become the leading cause of
hospital acquired infections in the US. Repurposing Food and Drug Administration (FDA) …

Reflecting the known biological activity of isoniazid-based hydrazones, seventeen
hydrazones of 4-(trifluoromethyl) benzohydrazide as their bioisosters were synthesized from …

Abstract Twenty-four 2-(4-oxo-2-thioxothiazolidin-3-yl) acetic acid (rhodanine-3-acetic acid)-
based amides, esters and 5-arylalkylidene derivatives were synthesized, characterized and …

Mycobacterium tuberculosis is an intracellular pathogen and the uptake of the
antimycobacterial compounds by host cells is limited. Novel antimycobacterials effective …

In this study, a series of twenty-two ring-substituted 6-hydroxynaphthalene-2-carboxanilides
was prepared and characterized. Primary in vitro screening of the synthesized compounds …

The research of innovative antimicrobial agents represents a cutting edge topic. Hence, we
synthesized and characterised novel salicylanilide N-monosubstituted carbamates. Twenty …

Salicylanilides have proved their activity against tuberculosis (TB). One weak electron-
withdrawing substituent is favored at the salicylic part, specially Cl or Br atoms at positions 4 …

The research of novel antimycobacterial drugs represents a cutting-edge topic. Thirty
phenolic N-monosubstituted carbamates, derivatives of salicylanilides and 4-chlorophenol …