[PDF][PDF] Pyrazoline derivatives: a worthy insight into the recent advances and potential pharmacological activities

MA Rahman, AA Siddiqui - Int J Pharm Sci Drug Res, 2010 - researchgate.net
Pyrazolines display a broad spectrum of potential pharmacological activities and are present
in a number of pharmacologically active molecules such as phenazone/amidopyrene …

In Melting Points We Trust: A Review on the Misguiding Characterization of Multicomponent Reactions Adducts and Intermediates

BAD Neto, PS Beck, JEP Sorto, MN Eberlin - Molecules, 2022 - mdpi.com
We discuss herein the problems associated with using melting points to characterize
multicomponent reactions'(MCRs) products and intermediates. Although surprising, it is not …

Synthesis, characterization, antibacterial and antioxidant studies of some heterocyclic compounds from triazole‐linked chalcone derivatives

R Santosh, MK Selvam, SU Kanekar… - …, 2018 - Wiley Online Library
In the current study, an efficient synthesis of new triazole‐linked chalcone 3 a‐g scaffold was
performed by multistep reaction sequence and was screened for their antibacterial activity …

Curcumin Derivatives as Potential Mosquito Larvicidal Agents against Two Mosquito Vectors, Culex pipiens and Aedes albopictus

D Matiadis, PGV Liggri, E Kritsi, N Tzioumaki… - International Journal of …, 2021 - mdpi.com
Vector-borne diseases have appeared or re-emerged in many Southern Europe countries
making the transmission of infectious diseases by mosquitoes (vectors) one of the greatest …

Design, synthesis and exploring the quantitative structure–activity relationship of some antioxidant flavonoid analogues

S Das, I Mitra, S Batuta, MN Alam, K Roy… - Bioorganic & medicinal …, 2014 - Elsevier
A series of flavonoid analogues were synthesized and screened for the in vitro antioxidant
activity through their ability to quench 1, 1-diphenyl-2-picryl hydrazyl (DPPH) radical. The …

Iron-facilitated oxidative radical decarboxylative cross-coupling between α-oxocarboxylic acids and acrylic acids: an approach to α, β-unsaturated carbonyls

Q Jiang, J Jia, B Xu, A Zhao… - The Journal of Organic …, 2015 - ACS Publications
The first Fe-facilitated decarboxylative cross-coupling reaction between α-oxocarboxylic
acids and acrylic acids in aqueous solution has been developed. This transformation is …

Carbon–carbon bond formation in acid deep eutectic solvent: chalcones synthesis via Claisen–Schmidt reaction

M Tiecco, R Germani, F Cardellini - RSC advances, 2016 - pubs.rsc.org
One of the most studied properties of novel organic solvents is represented by their use as
media for many chemical reactions. In this field Ionic Liquids (ILs) and more recently Deep …

Antioxidant, antimicrobial, cytotoxicity, and larvicidal activities of selected synthetic bis-chalcones

AM Kuttithodi, D Nikhitha, J Jacob, A Narayanankutty… - Molecules, 2022 - mdpi.com
Plants are known to have numerous phytochemicals and other secondary metabolites with
numerous pharmacological and biological properties. Among the various compounds …

Polyphenols bearing cinnamaldehyde scaffold showing cell growth inhibitory effects on the cisplatin-resistant A2780/Cis ovarian cancer cells

SY Shin, H Jung, S Ahn, D Hwang, H Yoon… - Bioorganic & medicinal …, 2014 - Elsevier
Ovarian carcinoma remains the most lethal among gynecological cancers. Chemoresistance
is a clinical problem that severely limits treatment success. To identify potent anticancer …

Larvicidal activity of substituted chalcones against Aedes aegypti (Diptera: Culicidae) and non‐target organisms

SK Targanski, JR Sousa, GMS de Pádua… - Pest management …, 2021 - Wiley Online Library
BACKGROUND The expansion of Aedes aegypti (Diptera: Culicidae) population has
increased the number of cases of arboviruses, in part due to the inefficiency and toxicity of …