Amide bond formation strategies: Latest advances on a dateless transformation

E Massolo, M Pirola, M Benaglia - European Journal of Organic …, 2020 - Wiley Online Library
The synthesis of amides remains one of the most important transformations and it is one of
the more frequently performed reactions. In the pharmaceutical industry, the formation of the …

Recent developments in catalytic amide bond formation

M Todorovic, DM Perrin - Peptide Science, 2020 - Wiley Online Library
Amide bond forming reactions are critical for both polypeptide synthesis and medicinal
chemistry. Most current approaches for amidation employ stoichiometric activating agents …

Direct catalytic amidations from carboxylic acid and ester derivatives: A review

A Taussat, RM de Figueiredo, JM Campagne - Catalysts, 2023 - mdpi.com
The prevalence of amides in biological systems and chemical fields such as polymers,
materials and natural products drives continuous research on novel procedures to obtain …

Sustainable amidation reactions–recent advances

AS Santos, AMS Silva… - European Journal of …, 2020 - Wiley Online Library
Due to the widespread occurrence of amides in modern pharmaceuticals and biologically
active compounds, amidation reaction is one of the most important reactions in organic …

Synthetic cinnamides and cinnamates: antimicrobial activity, mechanism of action, and in silico study

MC de Morais, E de Oliveira Lima, Y Perez-Castillo… - Molecules, 2023 - mdpi.com
The severity of infectious diseases associated with the resistance of microorganisms to
drugs highlights the importance of investigating bioactive compounds with antimicrobial …

Dulcisenes CE, polyoxygenated cyclohexenes, from Uvaria dulcis dunal and their cytotoxic activity

P Pailee, P Ploypradith, C Mahidol, S Ruchirawat… - Phytochemistry, 2022 - Elsevier
Dulcisenes CE, undescribed polyoxygenated cyclohexenes and twenty-one known
compounds were isolated from the dichloromethane extract of the leaves of Uvaria dulcis …

Antileishmanial Activity of Cinnamic Acid Derivatives against Leishmania infantum

MC de Morais, GA Medeiros, FS Almeida, JC Rocha… - Molecules, 2023 - mdpi.com
Leishmania infantum is the etiological agent of visceral leishmaniasis (VL) in South America,
the Mediterranean basin, and West and Central Asia. The most affected country, Brazil …

[HTML][HTML] Flow and On-Water Synthesis and Cancer Cell Cytotoxicity of Caffeic Acid Phenethyl Amide (CAPA) Derivatives

A Saucedo, M Subbarao, M Jemal… - International Journal of …, 2024 - mdpi.com
Caffeic acid phenethyl ester (CAPE) is a phenolic natural product with a wide range of
biological activities, including anticancer activity; however, the ester group of CAPE is …

[PDF][PDF] Cinnamates: Antimicrobial Activity, Mechanism of Action, and

MC Morais, EO Lima, Y Perez-Castillo, DPSC Sousa - Molecules, 2023 - academia.edu
The severity of infectious diseases associated with the resistance of microorganisms to
drugs highlights the importance of investigating bioactive compounds with antimicrobial …