Use of Lawesson's reagent in organic syntheses

T Ozturk, E Ertas, O Mert - Chemical reviews, 2007 - ACS Publications
Transformation of a carbonyl functional group into thiocarbonyl has been an important
interest to synthetic organic chemists for many years. Two reagents, phosphorus …

Synthesis of 3, 4, 5-Trisubstituted-1, 2, 4-triazoles

A Moulin, M Bibian, AL Blayo, S El Habnouni… - Chemical …, 2010 - ACS Publications
Triazoles are an important class of heterocyclic compounds not only as a core scaffold but
also as a benzo-fused (triazolopyridines and triazolopyrazines are well-known examples) or …

One-pot synthesis of 3, 4, 5-trisubstituted 1, 2, 4-triazoles via the addition of hydrazides to activated secondary amides

WS Bechara, IS Khazhieva, E Rodriguez… - Organic …, 2015 - ACS Publications
A general approach has been developed for the one-pot synthesis of 3, 4, 5-trisubstituted 1,
2, 4-triazoles from secondary amides and hydrazides via triflic anhydride activation followed …

Nitrogen-containing six-membered heterocycles: solid-phase synthesis

N Kaur, D Kishore - Synthetic Communications, 2014 - Taylor & Francis
Solid-phase organic synthesis is a rapidly expanding area of synthetic chemistry that is
being widely exploited in the search for new medicinally important compounds using …

Solution and solid-supported synthesis of 3, 4, 5-trisubstituted 1, 2, 4-triazole-based peptidomimetics

D Boeglin, S Cantel, A Heitz, J Martinez… - Organic letters, 2003 - ACS Publications
3, 4, 5-Trisubstituted 1, 2, 4-triazoles were synthesized in solution from various thioamides
and hydrazides in smooth experimental conditions leading to peptidomimetic scaffolds. This …

Trifluoromethylated 4,5-Dihydro-1,2,4-triazin-6(1H)-ones via (3+3)-Annulation of Nitrile Imines with α-Amino Esters

A Kowalczyk, K Świątek, M Celeda, G Utecht-Jarzyńska… - Materials, 2023 - mdpi.com
The synthesis of two series of monocyclic and bicyclic trifluoromethylated 4, 5-dihydro-1, 2, 4-
triazin-6 (1 H)-one derivatives based on (3+ 3)-annulation of methyl esters derived from …

Comprehensive survey of combinatorial library synthesis: 2003

RE Dolle - Journal of combinatorial chemistry, 2004 - ACS Publications
This is the seventh comprehensive survey in an ongoing annual review series in
combinatorial chemistry. 1 The format remains largely the same as in past years with …

Synthesis and reactions of 4‐benzoyl‐1,5‐diaryl‐1H‐pyrazole‐3‐carbonyl chlorides with various semi‐ and thiosemicarbazides

E Korkusuz, I Yıldırım - Journal of Heterocyclic Chemistry, 2010 - Wiley Online Library
Abstract The 1H‐pyrazole‐3‐carboxylic acids 2 were converted via reactions of their acid
chlorides 3 with some semi‐and thiosemicarbazide derivatives into the corresponding new …

Solid‐Supported Synthesis and 5‐HT7/5‐HT1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5‐dihydro‐1,2,4‐triazine‐6‐(1H)‐one

K Grychowska, N Masurier, P Verdié… - Chemical Biology & …, 2015 - Wiley Online Library
A series of arylpiperazinylbutyl derivatives of 4, 5‐dihydro‐1, 2, 4‐triazine‐6 (1H)‐ones was
designed and synthesized according to the new solid‐supported methodology. In this …

On the Reactions of Furan‐2,3‐diones with Oxindole (=1,3‐Dihydro‐2H‐indol‐2‐one) and Lawesson Reagent. Synthesis of New 1,3‐Dihydro‐2H‐indol‐2‐ones …

E Korkusuz, İ Yıldırım - Helvetica Chimica Acta, 2011 - Wiley Online Library
Lactone analogues of 3‐substituted oxindoles (= 1, 3‐dihydro‐2H‐indol‐2‐ones) and
nonbenzoid oxa‐analogous isoindigoid or nonbenzoid isoindigoid dyes were prepared by …