Triazoles are important five-membered heterocyclic scaffold due to their extensive biological
activities. This framework can be readily obtained in good to excellent yields on the …

Triazoles find applications in several major technological areas, and especially in drug
discovery. The click-chemistry approaches based on Huisgen's cycloaddition reaction are …

The 5‐heterofunctionalized triazoles are important scaffolds in bioactive compounds, but
current click reactions (CuAAC) cannot produce these core structures. A copper (I) …

A p-TsOH-mediated 1, 3-dipolar cycloaddition of nitroolefins and sodium azide for the
synthesis of 4-aryl-NH-1, 2, 3-triazoles has been developed. p-TsOH was discovered as a …

Copper (I)-catalyzed azide–alkyne cycloaddition (CuAAC) is an essential “click chemistry”
reaction that is widely used in chemical biology, medicinal chemistry and materials science …

The present feature article describes the different organocatalytic routes for the synthesis of
substituted 1, 2, 3-triazoles. This methodology has recently gained much attention due to its …

An overview of the latest developments in the metal-free synthesis of non-benzo-fused N-
functionalized and NH-1, 2, 3-triazoles is provided in this feature article. Synthetic studies …

Given the wide utility of click-chemistry reactions for the preparation of simple moieties within
large architecturally complex materials, this minireview article aims at surveying papers …

Metal-free 1, 3-dipolar cycloaddition reactions have proven to be a powerful tool for the
assembly of key heterocycles, in particular diversely functionalized 1, 2, 3-triazoles. A …

The domino reactions between NH-based secondary enaminones and tosyl azide have
been developed for the synthesis of various N-substituted 1, 2, 3-triazoles by employing t …