Review on therapeutic potential of peptides: Advancements in synthesis methods, linear and cyclic peptides, and strategies for overcoming challenges

N Lalani, S Tivari, V Jain, Y Jadeja - Peptide Science, 2024 - Wiley Online Library
In the realm of therapeutic peptides, tremendous progress has been achieved in the last two
decades. The building block of peptides that is,'Amino Acid'has been modified by various …

Design, Synthesis, and Evaluation of Quinoline‐1,2,3‐Triazole Hybrids as CYP51 Inhibitors: In Silico Study and In Vitro Antimicrobial Assessment

BK Chabhadiya, HN Naik, BA Mohite, I Ahmad… - …, 2024 - Wiley Online Library
Novel Quinoline‐triazole hybrid derivatives (9 a–9 l) were designed and synthesized via
click reaction methodology to develop lead compounds with good antibacterial and …

[HTML][HTML] Synthesis and Antifungal Activity of Fmoc-Protected 1,2,4-Triazolyl-α-Amino Acids and Their Dipeptides Against Aspergillus Species

T Sargsyan, L Stepanyan, H Panosyan, H Hakobyan… - Biomolecules, 2025 - mdpi.com
In recent years, fungal infections have emerged as a significant health concern across
veterinary species, especially in livestock such as cattle, where fungal diseases can result in …

Synthesis, characterization, biological activities, and computational studies of pyrazolyl–thiazole derivatives of thiophene

SK Bhagwat, TJ Pawar, SA Kulkarni, AA Patil… - RSC …, 2024 - pubs.rsc.org
This study reports the synthesis, characterization, and biological evaluation of a series of
pyrazolyl–thiazole derivatives of thiophene. Seven compounds were synthesized and …