Biological activity of oxadiazole and thiadiazole derivatives

UA Atmaram, SM Roopan - Applied Microbiology and Biotechnology, 2022 - Springer
The 5-membered oxadiazole and thiadiazole scaffolds are the most privileged and well-
known heterocycles, being a common and essential feature of a variety of natural products …

1, 3, 4-Thiadiazole: synthesis, reactions, and applications in medicinal, agricultural, and materials chemistry

Y Hu, CY Li, XM Wang, YH Yang, HL Zhu - Chemical reviews, 2014 - ACS Publications
Over the past decades, the bulk of chemists' interests have been on heterocyclic compounds
and their various derivatives as well as their applications in the pharmaceutical and …

Synthesis and antimicrobial activity of some new pyrimidinone and oxazinone derivatives fused with thiophene rings using 2-chloro-6-ethoxy-4-acetylpyridine as …

ASM Hossan, HMA Abu-Melha, MA Al-Omar… - Molecules, 2012 - mdpi.com
A series of pyridines, pyrimidinones, oxazinones and their derivatives were synthesized as
antimicrobial agents using citrazinic acid (2, 6-dihydroxyisonicotinic acid) as a starting …

Synthesis and Anticancer Properties of Silver (I) Complexes Containing 2, 6‐Bis (substituted) pyridine Derivatives

KA Ali, MM Abd-Elzaher… - International Journal of …, 2013 - Wiley Online Library
Several new 2, 6‐bis (substituted) pyridine ligands and 2, 6‐bis (substituted) pyridine Ag (I)
nitrate complexes were synthesized and characterized spectroscopically. The newly …

A metal-free tandem approach to prepare structurally diverse N-heterocycles: synthesis of 1, 2, 4-oxadiazoles and pyrimidinones

PK Gupta, MK Hussain, M Asad, R Kant… - New Journal of …, 2014 - pubs.rsc.org
A metal-free one-pot approach to the diversity oriented synthesis of N-heterocycles, 1, 2, 4-
oxadiazoles and 2, 6 disubstituted pyrimidin-4-ones is described via carboxamidation of …

Straightforward synthesis of novel substituted 1, 3, 4-thiadiazole derivatives in choline chloride-based deep eutectic solvent

SM Shahcheragh, A Habibi, S Khosravi - Tetrahedron Letters, 2017 - Elsevier
A one-pot, three-component route for the synthesis of novel 1, 3, 4-thiadiazole derivatives
using a ketene S, S-acetal, a carbonyl compound and thiocarbohydrazide is described. The …

Synthesis of novel tripeptides based on dibenzofuran-2-sulfonyl-[aromatic and hydroxy aromatic residues]: Towards antimicrobial and antifungal agents

HSA Al-Salem, AM Naglah… - Journal of …, 2017 - ingentaconnect.com
A series of linear tripeptide derivatives (4–29) have been prepared and evaluated as
antimicrobial agents via the synthesis of dibenzofuran-2-sulfonyl chloride (3). The …

Structural Investigation and Hirshfeld Surface Analysis of N-(3-Chloro-4-Methylphenyl)-2-(3-Nitrobenzamido)Benzamide

MM Ayoob, FE Hawaiz, N Dege, S Kansız - Journal of Structural Chemistry, 2023 - Springer
A new synthesis of N-(3-chloro-4-methylphenyl)-2-(3-nitrobenzamido) benzamide was
developed in acetic acid as a solvent using the reaction of 3-choloro-4-methylaniline, and 2 …

A highly selective and sensitive reusable colorimetric sensor for Ag+ based on thiadiazole-functionalized polyacrylonitrile fiber

R Gao, G Xu, L Zheng, Y Xie, M Tao… - Journal of Materials …, 2016 - pubs.rsc.org
A thiadiazole-functionalized polyacrylonitrile fiber (DPTD-PANPF) qualitative colorimetric
sensor was prepared for the first time, and its absorption properties were investigated in …

HIV-1 and HSV-1 virus activities of some new polycyclic nucleoside pyrene candidates

NM Khalifa, MA Al-Omar, AEGE Amr… - International journal of …, 2013 - Elsevier
In continuation of our previous work, a novel series of polycyclic derivatives 2–8
incorporated heterocyclic and sugar moieties were synthesized by using pyren-1-aldehyde …