Synthesis of covalent organic frameworks via Kabachnik-Fields reaction for water treatment

WX Wu, F Li, BJ Yao, LG Ding, JL Kan, F Liu… - Journal of Hazardous …, 2022 - Elsevier
Providing safe and clean domestic water for people is currently one of the greatest
worldwide issues. In this context, heavy metal ions and pathogenic microbes are the two …

Design, synthesis and evaluation of pyrazole bearing α-aminophosphonate derivatives as potential acetylcholinesterase inhibitors against Alzheimer's disease

S Shaikh, P Dhavan, G Pavale, MMV Ramana… - Bioorganic …, 2020 - Elsevier
A series of novel scaffold of N-substituted pyrazole derived α-aminophosphonates were
designed, synthesized and evaluated for their anti-cholinesterase activity. Porcine …

Chromone containing hybrid analogs: Synthesis and applications in medicinal chemistry

PS Auti, S Jagetiya, AT Paul - Chemistry & Biodiversity, 2023 - Wiley Online Library
The use of privileged scaffolds has proven beneficial for generating novel bioactive scaffolds
in drug discovery program. Chromone is one such privileged scaffold that has been …

Recent Advances in the Synthesis of Dialkyl (Aryl) α-(Aryl/Heterocyclic/Heteroaryl-α-(Aryl/Heteroarylamino) Phosphonates

TE Ali, MA Assiri, M Hussien… - Current Organic …, 2023 - ingentaconnect.com
This review describes recent advances that are commonly applied in the synthesis of dialkyl
(aryl) α-aminophosphonates containing heterocyclic compounds. The target structures are …

Design, synthesis and evaluation of new chromone-derived aminophosphonates as potential acetylcholinesterase inhibitor

S Shaikh, P Dhavan, MMV Ramana, BL Jadhav - Molecular Diversity, 2021 - Springer
A series of novel N-substituted α-aminophosphonates-bearing chromone moiety were
synthesized and evaluated for acetylcholinesterase (AChE), butyrylcholinesterase (BuChE) …

Design, synthesis, molecular modeling, and biological evaluation of novel α-aminophosphonates based quinazolinone moiety as potential anticancer agents: DFT …

MK Awad, MF Abdel-Aal, FM Atlam, HA Hekal - Journal of Molecular …, 2018 - Elsevier
Abstract Diphenyl (aryl)(4-oxo-2-phenyl-4H-quinazolin-3-yl)-acetic acid hydrazino methyl
phosphonate (IIIa-k) was achieved upon the reaction of 3, 4-dihydro-(4-oxo-2-phenyl-4H …

Green approach to the synthesis of α-aminophosphonate-tetrahydroisoquinoline hybrids and their anti-cholinesterase activity

J Marchán-García, E Buxaderas, DN Stratico… - Bioorganic …, 2024 - Elsevier
A series of 19 novel α-aminophosphonate-tetrahydroisoquinoline hybrids were synthesized
through a cross dehydrogenative coupling reaction between N-aryl-tetrahydroisoquinolines …

Design, synthesis and biological evaluation of novel antipyrine based α-aminophosphonates as anti-Alzheimer and anti-inflammatory agent

S Shaikh, P Dhavan, P Singh, J Uparkar… - Journal of …, 2023 - Taylor & Francis
Herein, a series of novel antipyrine based α-aminophosphonates derivatives were
synthesized and characterized. The synthesized derivatives were subjected for in vitro …

Promiscuous lipase catalyzed a new P–C bond formation: Green and efficient protocol for one‐pot synthesis of α‐aminophosphonates

S Guezane‐Lakoud, M Toffano… - Heteroatom …, 2017 - Wiley Online Library
Abstract α‐Aminophosphonates are valuable substructures with important biological and
pharmacological properties. Lipase catalytic promiscuity is a new method in the organic …

Synthesis carbonic anhydrase enzyme inhibition and antioxidant activity of novel benzothiazole derivatives incorporating glycine, methionine, alanine, and …

DÜ Payaz, FZ Küçükbay, H Küçükbay… - Journal of enzyme …, 2019 - Taylor & Francis
Thirteen novel benzothiazole derivatives incorporating glycine, methionine, alanine, and
phenylalanine were synthesised by facile acylation reactions through benzotriazole or DCC …