Hydrazide–hydrazones as potential antimicrobial agents: overview of the literature since 2010
Ł Popiołek - Medicinal Chemistry Research, 2017 - Springer
Hydrazide–hydrazone derivatives are present in many bioactive molecules and display a
wide variety of biological activities, such as antibacterial, antitubercular, antifungal …
wide variety of biological activities, such as antibacterial, antitubercular, antifungal …
Synthesis, spectroscopic properties and antipathogenic activity of new thiourea derivatives
C Limban, L Marutescu, MC Chifiriuc - Molecules, 2011 - mdpi.com
A number of acylthioureas, 2-((4-methylphenoxy) methyl)-N-(aryl-carbamothioyl)
benzamides (aryl= 3, 5-dichlorophenyl, 2, 3-dichlorophenyl, 3, 4-dichloro-phenyl, 2, 4, 5 …
benzamides (aryl= 3, 5-dichlorophenyl, 2, 3-dichlorophenyl, 3, 4-dichloro-phenyl, 2, 4, 5 …
Synthesis, X-ray, Hirshfeld surface analysis, exploration of DNA binding, urease enzyme inhibition and anticancer activities of novel adamantane-naphthyl thiourea …
(adamantane-1-carbonyl-3-(1-naphthyl)) thiourea (C 22 H 24 N 2 OS (4), was synthesized
by the reaction of freshly prepared adamantane-1-carbonyl chloride from corresponding …
by the reaction of freshly prepared adamantane-1-carbonyl chloride from corresponding …
[HTML][HTML] Design, synthesis, and molecular docking studies of a conjugated thiadiazole–thiourea scaffold as antituberculosis agents
Design, Synthesis, and Molecular Docking Studies of a Conjugated Thiadiazole–Thiourea
Scaffold as Antituberculosis Agents Toggle navigation J-STAGE home Browse All titles All …
Scaffold as Antituberculosis Agents Toggle navigation J-STAGE home Browse All titles All …
Synthesis, anticancer activity, toxicity evaluation and molecular docking studies of novel phenylaminopyrimidine—(thio) urea hybrids as potential kinase inhibitors
Thirty-two novel urea/thiourea compounds as potential kinase inhibitor were designed,
synthesized and evaluated for their cytotoxic activity on breast (MCF7), colon (HCT116) and …
synthesized and evaluated for their cytotoxic activity on breast (MCF7), colon (HCT116) and …
[HTML][HTML] Synthesis and antiproliferative screening of novel doubly modified colchicines containing urea, thiourea and guanidine moieties
J Krzywik, E Maj, A Nasulewicz-Goldeman… - Bioorganic & Medicinal …, 2021 - Elsevier
A new series of 10-demethoxy-10-methylaminocolchicines bearing urea, thiourea or a
guanidine moieties at position C7 has been designed, synthesized and evaluated for in vitro …
guanidine moieties at position C7 has been designed, synthesized and evaluated for in vitro …
Benzocaine as a precursor of promising derivatives: Synthesis, reactions, and biological activity
Electrophilic and nucleophilic reactions of benzocaine are the most common procedures to
construct a library of benzocaine derivatives, which have promising features that could be …
construct a library of benzocaine derivatives, which have promising features that could be …
Amido-Schiff base derivatives as colorimetric fluoride sensor: effect of nitro substitution on the sensitivity and color change
A series of Schiff bases synthesized by the condensation of benzohydrazide and–NO 2
substituted benzaldehyde have been used as selective fluoride ion sensor. Test paper …
substituted benzaldehyde have been used as selective fluoride ion sensor. Test paper …
Design and Synthesis of N-Arylphthalimides as Inhibitors of Glucocorticoid-Induced TNF Receptor-Related Protein, Proinflammatory Mediators, and Cytokines in …
N-Arylphthalimides (1–10P) derived from thalidomide by insertion of hydrophobic groups
were evaluated for anti-inflammatory activity, and (4-(1, 3-dioxo-1, 3-dihydro-2 H-isoindol-2 …
were evaluated for anti-inflammatory activity, and (4-(1, 3-dioxo-1, 3-dihydro-2 H-isoindol-2 …
Novel thiourea derivatives against Mycobacterium tuberculosis: synthesis, characterization and molecular docking studies
Abstract N-((2-chloropyridin-3-yl) carbamothioyl) thiophene-2-carboxamide (HL1), N-((6-
methylpyridin-2-yl) carbamothioyl) thiophene-2-carboxamide (HL2), N-(allylcarbamothioyl) …
methylpyridin-2-yl) carbamothioyl) thiophene-2-carboxamide (HL2), N-(allylcarbamothioyl) …